| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3614381 | B | Inhibition of human FAAH expressed in COS7 cell membranes at 10 uM pre-incubated for 10 mins before [3H]-AEA substrate addition by liquid scintillation counting | Homo sapiens | 26 | ALA3612019 | cell-based format | Scientific Literature | |
| 2. | ALA3614383 | B | Inhibition of human FAAH expressed in COS7 cell membranes at 20 uM pre-incubated for 10 mins before [3H]-AEA substrate addition by liquid scintillation counting | Homo sapiens | 1 | ALA3612019 | cell-based format | Scientific Literature | |
| 3. | ALA3614384 | B | Inhibition of human MAGL expressed in HEK293 cells at 10 uM pre-incubated for 10 mins before 2-AG substrate addition by HPLC method | Homo sapiens | 29 | ALA3612019 | cell-based format | Scientific Literature | |
| 4. | ALA3614386 | B | Inhibition of human MAGL expressed in HEK293 cells at 20 uM pre-incubated for 10 mins before 2-AG substrate addition by HPLC method | Homo sapiens | 1 | ALA3612019 | cell-based format | Scientific Literature | |
| 5. | ALA3614931 | B | Inhibition of human ABHD6 expressed in HEK293 cells assessed as reduction in glycerol production from 1-AG hydrolysis pre-incubated for 30 mins before 1-AG substrate addition and measured 90 mins post substrate addition by fluorescence method | Homo sapiens | 7 | ALA3612019 | cell-based format | Scientific Literature | |
| 6. | ALA3614932 | B | Selectivity for human ABHD6 expressed in HEK293 cells over human FAAH expressed in COS7 cell membranes | Homo sapiens | 1 | ALA3612019 | cell-based format | Scientific Literature | |
| 7. | ALA3614933 | B | Selectivity for human ABHD6 expressed in HEK293 cells over human MAGL expressed in COS7 cell membranes | Homo sapiens | 1 | ALA3612019 | cell-based format | Scientific Literature | |
| 8. | ALA3614934 | B | Inhibition of ABHD6 in mouse whole brain membranes at 10 uM incubated for 1 hr by TAMRA-FP probe based competitive activity-based protein profiling assay | Mus musculus | 1 | ALA3612019 | cell membrane format | Scientific Literature | |
| 9. | ALA3614935 | B | Inhibition of FAAH in mouse whole brain membranes at 10 uM incubated for 1 hr by TAMRA-FP probe based competitive activity-based protein profiling assay | Mus musculus | 2 | ALA3612019 | cell membrane format | Scientific Literature | |
| 10. | ALA3614936 | B | Inhibition of MAGL in mouse whole brain membranes at 10 uM incubated for 1 hr by TAMRA-FP probe based competitive activity-based protein profiling assay | Mus musculus | 2 | ALA3612019 | cell membrane format | Scientific Literature | |
| 11. | ALA3614937 | B | Inhibition of ABHD12 in mouse whole brain membranes at 10 uM incubated for 1 hr by TAMRA-FP probe based competitive activity-based protein profiling assay | Mus musculus | 2 | ALA3612019 | cell membrane format | Scientific Literature | |
| 12. | ALA3614939 | B | Inhibition of FAAH in mouse whole brain membranes at 32.5 uM incubated for 1 hr by TAMRA-FP probe based competitive activity-based protein profiling assay | Mus musculus | 1 | ALA3612019 | cell membrane format | Scientific Literature | |
| 13. | ALA3614940 | B | Inhibition of MAGL in mouse whole brain membranes at 32.5 uM incubated for 1 hr by TAMRA-FP probe based competitive activity-based protein profiling assay | Mus musculus | 1 | ALA3612019 | cell membrane format | Scientific Literature | |
| 14. | ALA3614941 | B | Inhibition of ABHD12 in mouse whole brain membranes at 32.5 uM incubated for 1 hr by TAMRA-FP probe based competitive activity-based protein profiling assay | Mus musculus | 1 | ALA3612019 | cell membrane format | Scientific Literature | |
| 15. | ALA3614942 | F | Agonist activity at CB1R in rat cerebellar membranes at 10 uM by [35S]GTPgammaS binding assay | Rattus norvegicus | 1 | ALA3612019 | cell membrane format | Scientific Literature | |
| 16. | ALA3614944 | F | Agonist activity at human CB2R expressed in CHO cell membranes at 10 uM by [35S]GTPgammaS binding assay | Homo sapiens | 1 | ALA3612019 | cell-based format | Scientific Literature | |
| 17. | ALA3614947 | F | Antagonist activity at CB1R in rat cerebellar membranes assessed as inhibition of HU210-induced response at 10 uM by [35S]GTPgammaS binding assay | Rattus norvegicus | 1 | ALA3612019 | cell membrane format | Scientific Literature | |
| 18. | ALA3614949 | B | Inhibition of human ABHD6 expressed in HEK293 cells at 1 uM pre-incubated for 10 mins before 2-AG substrate addition followed by rapid 40 fold compound dilution measured after 10 mins by HPLC method | Homo sapiens | 3 | ALA3612019 | cell-based format | Scientific Literature | |
| 19. | ALA3614950 | B | Inhibition of human ABHD6 expressed in HEK293 cells at 1 uM pre-incubated for 10 mins before 2-AG substrate addition followed by rapid 40 fold compound dilution measured after 30 mins by HPLC method | Homo sapiens | 3 | ALA3612019 | cell-based format | Scientific Literature | |
| 20. | ALA3614951 | B | Inhibition of human ABHD6 expressed in HEK293 cells at 1 uM pre-incubated for 10 mins before 2-AG substrate addition followed by rapid 40 fold compound dilution measured after 60 mins by HPLC method | Homo sapiens | 3 | ALA3612019 | cell-based format | Scientific Literature |
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