| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3616091 | B | Inhibition of MGAT3 (unknown origin) assessed effect on incorporation of [1-14C]decanoyl moiety into triacylglycerol using [1-14C]decanoyl-CoA and 1,2-didecanoyl-sn-glycerol as substrates pre-incubated for 30 mins before substrate addition | Homo sapiens | 10 | ALA3612040 | single protein format | Scientific Literature | |
| 2. | ALA3616240 | B | Inhibition of MGAT1 (unknown origin) assessed as effect on incorporation of [1-14C]decanoyl moiety into DAG using [1-14C]decanoyl-CoA and 2-oleoylglycerol as substrates | Homo sapiens | 2 | ALA3612040 | single protein format | Scientific Literature | |
| 3. | ALA3616241 | B | Inhibition of MGAT2 (unknown origin) assessed as effect on incorporation of [1-14C]decanoyl moiety into DAG using [1-14C]decanoyl-CoA and 1-decanoyl-rac-glycerol as substrates | Homo sapiens | 2 | ALA3612040 | single protein format | Scientific Literature | |
| 4. | ALA3616242 | B | Inhibition of DGAT1 (unknown origin) assessed as effect on incorporation of [1-14C]decanoyl moiety into TG using [1-14C]decanoyl-CoA and 1,2-didecanoyl-sn-glycerol as substrates | Homo sapiens | 2 | ALA3612040 | single protein format | Scientific Literature | |
| 5. | ALA3616243 | B | Inhibition of DGAT2 (unknown origin) using [1-14C]decanoyl-CoA and didecanoyl-sn-glycerol substrates incubated for 40 mins | Homo sapiens | 2 | ALA3612040 | single protein format | Scientific Literature | |
| 6. | ALA3616244 | P | Lipophilicity, logD of the compound at pH 7.4 | 10 | ALA3612040 | small-molecule physicochemical format | Scientific Literature | ||
| 7. | ALA3616245 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 10 | ALA3612040 | assay format | Scientific Literature | |
| 8. | ALA3616246 | A | Apparent permeability in RRCK cells | Canis lupus familiaris | 10 | ALA3612040 | cell-based format | Scientific Literature | |
| 9. | ALA3616247 | A | Inhibition of CYP2C8 (unknown origin) at 3 uM | Homo sapiens | 3 | ALA3612040 | single protein format | Scientific Literature | |
| 10. | ALA3616248 | A | Inhibition of CYP2C9 (unknown origin) at 3 uM | Homo sapiens | 3 | ALA3612040 | single protein format | Scientific Literature |
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