| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3624059 | B | Inhibition of recombinant human ADAMTS4 (213 to 575 amino acid residues) using WAAG-3R as substrate preincubated for 15 mins followed by substrate addition measured every 30 secs for 1 hr | Homo sapiens | 33 | single protein format | Scientific Literature | ||
| 2. | ALA3624060 | B | Inhibition of ADAMTS5 (unknown origin) using WAAG-3R as substrate at 10 uM preincubated for 15 mins followed by substrate addition measured every 30 secs for 1 hr relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA3624061 | B | Inhibition of ADAMTS5 (unknown origin) using WAAG-3R as substrate preincubated for 15 mins followed by substrate addition measured every 30 secs for 1 hr | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA3624062 | B | Inhibition of human recombinant ADAMTS13 using FRETSVWF73 as substrate by fluorescence assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA3624063 | B | Inhibition of human recombinant MMP13 using 5-FAMTPGPLGL[Dap(DNP)]ARRK(5-TAMRA)-amide as substrate after 45 mins | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA3624064 | B | Inhibition of human recombinant TACE using Mca-PLAQAV-Dpa-RSSSR-NH2 as substrate preincubated for 15 mins measured every 30 secs for 30 mins by fluorescence assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA3624065 | B | Selectivity ratio of IC50 for ADAMTS5 (unknown origin) to IC50 for recombinant human ADAMTS4 (213 to 575 amino acid residues) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 8. | ALA3624066 | B | Selectivity ratio of IC50 for human recombinant ADAMTS13 to IC50 for recombinant human ADAMTS4 (213 to 575 amino acid residues) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA3624067 | B | Selectivity ratio of IC50 for human recombinant MMP13 to IC50 for recombinant human ADAMTS4 (213 to 575 amino acid residues) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA3624202 | B | Selectivity ratio of IC50 for human recombinant TACE to IC50 for recombinant human ADAMTS4 (213 to 575 amino acid residues) | Homo sapiens | 1 | assay format | Scientific Literature |
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