| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3626367 | B | Agonist activity at wild type AR expressed in human SC cells assessed as effect on cell proliferation by WST-8 assay | Homo sapiens | 30 | cell-based format | Scientific Literature | ||
| 2. | ALA3626368 | B | Antagonist activity at wild type AR expressed in human SC cells assessed as inhibition of 1 nM DHT-induced cell proliferation after 3 days by WST-8 assay | Homo sapiens | 30 | cell-based format | Scientific Literature | ||
| 3. | ALA3626369 | B | Antagonist activity at wild type AR expressed in human SC cells assessed as inhibition of 0.3 to 10 nM DHT-induced cell proliferation after 3 days by WST-8 assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 4. | ALA3626370 | B | Displacement of [3H]-DHT from human GST fused AR-LBD (627 to 919 amino acids) transfected in Escherichia coli HB 101 after 15 hrs by liquid scintillation counting assay | Homo sapiens | 7 | assay format | Scientific Literature | ||
| 5. | ALA3626371 | B | Antagonist activity at AR T877A mutant expressed in human LNCaP cells assessed as inhibition of 10 nM DHT-stimulated cell proliferation after 6 days by WST-8 assay | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 6. | ALA3626372 | B | Antagonist activity at AR T877A mutant expressed in human LNCaP cells assessed as inhibition of 10 nM testosterone-induced PSA production after 48 hrs by ELISA method | Homo sapiens | 7 | cell-based format | Scientific Literature | ||
| 7. | ALA3624442 | F | Cytotoxicity against androgen-independent human PC3 cells assessed as inhibition of cell proliferation after 3 days by WST-8 assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 8. | ALA5140935 | F | Antiproliferative activity against human LNCaP cells | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 9. | ALA5140965 | F | Antiproliferative activity against mouse SC-3 cells | Mus musculus | 3 | cell-based format | Scientific Literature | ||
| 10. | ALA5140966 | B | Antagonist activity at Androgen receptor in human LNCaP cells assessed as inhibition of PSA expression | Homo sapiens | 5 | cell-based format | Scientific Literature |
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