| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3627015 | B | Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1 hr after substrate addition by cell free kinase assay | Homo sapiens | 40 | ALA3621069 | single protein format | Scientific Literature | |
| 2. | ALA3627019 | B | Inhibition of SYK-mediated TNFalpha production in human IgG-stimulated human THP1 cells incubated for 18 hrs by ELISA method | Homo sapiens | 4 | ALA3621069 | cell-based format | Scientific Literature | |
| 3. | ALA3627020 | B | Inhibition of purified full-length human ZAP70 pre-incubated for 30 mins at room temperature before UlighTM-PolyGT peptide substrate addition and measured 1 hr after substrate addition by cell free kinase assay | Homo sapiens | 4 | ALA3621069 | single protein format | Scientific Literature | |
| 4. | ALA3627021 | B | Inhibition of human JAK2 pre-incubated for 30 mins at room temperature before substrate addition and measured 1 hr after substrate addition by cell free kinase assay | Homo sapiens | 4 | ALA3621069 | single protein format | Scientific Literature | |
| 5. | ALA3627022 | B | Inhibition of JAK3 (unknown origin) pre-incubated for 30 mins at room temperature before substrate addition and measured 1 hr after substrate addition by cell free kinase assay | Homo sapiens | 4 | ALA3621069 | single protein format | Scientific Literature | |
| 6. | ALA3627023 | B | Inhibition of Aurora B kinase (unknown origin) pre-incubated for 30 mins at room temperature before substrate addition and measured 1 hr after substrate addition by cell free kinase assay | Homo sapiens | 4 | ALA3621069 | single protein format | Scientific Literature | |
| 7. | ALA3627024 | B | Inhibition of KDR (unknown origin) pre-incubated for 30 mins at room temperature before substrate addition and measured 1 hr after substrate addition by cell free kinase assay | Homo sapiens | 4 | ALA3621069 | single protein format | Scientific Literature | |
| 8. | ALA3627025 | B | Inhibition of human RET pre-incubated for 30 mins at room temperature before substrate addition and measured 1 hr after substrate addition by cell free kinase assay | Homo sapiens | 4 | ALA3621069 | single protein format | Scientific Literature | |
| 9. | ALA3627026 | B | Inhibition of purified full-length human SYK at 0.1 uM pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1 hr after substrate addition by cell free kinase assay | Homo sapiens | 1 | ALA3621069 | single protein format | Scientific Literature | |
| 10. | ALA3627027 | B | Inhibition of purified full-length human SYK at 0.01 uM pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1 hr after substrate addition by cell free kinase assay | Homo sapiens | 1 | ALA3621069 | single protein format | Scientific Literature | |
| 11. | ALA3627063 | B | Inhibition of human MLK1 at 0.1 uM | Homo sapiens | 1 | ALA3621069 | single protein format | Scientific Literature | |
| 12. | ALA3627064 | B | Inhibition of human MLK1 at 0.01 uM | Homo sapiens | 1 | ALA3621069 | single protein format | Scientific Literature | |
| 13. | ALA3627065 | A | Stability in human liver microsomes | Homo sapiens | 3 | ALA3621069 | assay format | Scientific Literature | |
| 14. | ALA3627066 | A | Apparent permeability from apical to basolateral side in human Caco2 cells | Homo sapiens | 3 | ALA3621069 | cell-based format | Scientific Literature | |
| 15. | ALA3627067 | A | Apparent permeability from basolateral to apical side in human Caco2 cells | Homo sapiens | 3 | ALA3621069 | cell-based format | Scientific Literature | |
| 16. | ALA3627068 | A | Inhibition of CYP450 (unknown origin) | Homo sapiens | 3 | ALA3621069 | assay format | Scientific Literature | |
| 17. | ALA3627069 | A | Unbound fraction in human plasma | Homo sapiens | 3 | ALA3621069 | cell-free format | Scientific Literature | |
| 18. | ALA3627070 | B | Inhibition of human ERG by manual patch clamp assay | Homo sapiens | 3 | ALA3621069 | assay format | Scientific Literature | |
| 19. | ALA3627071 | T | Genotoxicity in Salmonella typhimurium TA98 at 5000 lg/plate in presence of liver S9 fraction by Ames test | Salmonella enterica subsp. enterica serovar Typhimurium | 3 | ALA3621069 | organism-based format | Scientific Literature | |
| 20. | ALA3627072 | T | Genotoxicity in Salmonella typhimurium TA98 at 5000 lg/plate in absence of liver S9 fraction by Ames test | Salmonella enterica subsp. enterica serovar Typhimurium | 3 | ALA3621069 | organism-based format | Scientific Literature |
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