#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA3624232	F	Antitumor activity against bicalutamide-resistant human CWR22 cells in Balb/c athymic (nu/nu) mouse CWR22-BMSLD1 prostate cancer xenograft model assessed as tumor growth inhibition at 90 mg/kg, po qd administered for 45 days measured for 10 days during compound dosing	Homo sapiens	1	ALA3621143	organism-based format	Scientific Literature
2.	ALA3624233	B	Displacement of [3H]-DHT from androgen receptor in human MDA-MB-453 cells after 90 mins by TopCount analysis	Homo sapiens	15	ALA3621143	cell-based format	Scientific Literature
3.	ALA3624234	B	Antagonist activity at androgen receptor in human MDA-MB-453 cells assessed as inhibition of DHT-induced PSA expression by alkaline phosphatase reporter gene assay	Homo sapiens	15	ALA3621143	cell-based format	Scientific Literature
4.	ALA3624369	F	In vivo antagonist activity at androgen receptor in immature Sprague-Dawley rat prostate weight model assessed as testosterone propionate-induced weight of seminal vesicles over full body weight at 1 mg/kg, po qd administered for 4 days	Rattus norvegicus	12	ALA3621143	organism-based format	Scientific Literature
5.	ALA3624801	F	In vivo antagonist activity at androgen receptor in immature Sprague-Dawley rat prostate weight model assessed as testosterone propionate-induced weight of seminal vesicles over full body weight at 10 mg/kg, po qd administered for 4 days	Rattus norvegicus	12	ALA3621143	organism-based format	Scientific Literature
6.	ALA3624802	A	Plasma concentration in immature Sprague-Dawley rat prostate weight model at 1 mg/kg, po qd administered for 4 days measured 2 hrs post last dose on day 4	Rattus norvegicus	12	ALA3621143	organism-based format	Scientific Literature
7.	ALA3624803	A	Plasma concentration in immature Sprague-Dawley rat prostate weight model at 10 mg/kg, po qd administered for 4 days measured 2 hrs post last dose on day 4	Rattus norvegicus	12	ALA3621143	organism-based format	Scientific Literature
8.	ALA3624805	A	Drug metabolism in mouse hepatocytes assessed per 10'6 cells	Mus musculus	1	ALA3621143	cell-based format	Scientific Literature
9.	ALA3624806	F	Cytotoxicity against human LNCAP cells	Homo sapiens	1	ALA3621143	cell-based format	Scientific Literature
10.	ALA3624807	A	Inhibition of human CYP1A2	Homo sapiens	1	ALA3621143	single protein format	Scientific Literature
11.	ALA3624808	A	Inhibition of human CYP2B6	Homo sapiens	1	ALA3621143	single protein format	Scientific Literature
12.	ALA3624809	A	Inhibition of human CYP2C8	Homo sapiens	1	ALA3621143	single protein format	Scientific Literature
13.	ALA3624810	A	Inhibition of human CYP2C9	Homo sapiens	1	ALA3621143	single protein format	Scientific Literature
14.	ALA3624811	A	Inhibition of human CYP2D6	Homo sapiens	1	ALA3621143	single protein format	Scientific Literature
15.	ALA3624812	A	Inhibition of human CYP3A4	Homo sapiens	1	ALA3621143	single protein format	Scientific Literature
16.	ALA3624813	A	Transactivation of human PXR	Homo sapiens	1	ALA3621143	single protein format	Scientific Literature
17.	ALA3624814	B	Inhibition of human ERG at 30 uM relative to control	Homo sapiens	1	ALA3621143	single protein format	Scientific Literature
18.	ALA3624815	A	Fraction unbound in mouse plasma by equilibrium dialysis method	Mus musculus	1	ALA3621143	cell-free format	Scientific Literature
19.	ALA3624816	A	Fraction unbound in rat plasma by equilibrium dialysis method	Rattus norvegicus	1	ALA3621143	cell-free format	Scientific Literature
20.	ALA3624817	A	Fraction unbound in dog plasma by equilibrium dialysis method	Canis lupus familiaris	1	ALA3621143	cell-free format	Scientific Literature