| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3636924 | B | Displacement of [3H]PK11195 from TSPO in human HEK293T cell membranes incubated for 90 mins by competition radioligand binding assay | Homo sapiens | 5 | ALA3632527 | cell-based format | Scientific Literature | |
| 2. | ALA3636925 | B | Displacement of [3H]PK11195 from TSPO in human T98G cell membranes incubated for 90 mins by competition radioligand binding assay | Homo sapiens | 5 | ALA3632527 | cell-based format | Scientific Literature | |
| 3. | ALA3636926 | F | Antiproliferative activity against human T98G cells at 1 to 100 uM incubated for 48 hrs by BrdU enzyme-linked immunosorbent assay | Homo sapiens | 5 | ALA3632527 | cell-based format | Scientific Literature | |
| 4. | ALA3636927 | F | Potentiation of antiproliferative activity of PK11195 against human T98G cells incubated for 48 hrs by BrdU enzyme-linked immunosorbent assay | Homo sapiens | 1 | ALA3632527 | cell-based format | Scientific Literature | |
| 5. | ALA3636928 | F | Potentiation of antiproliferative activity of PK11195 at 10 uM against human T98G cells incubated for 48 hrs by BrdU enzyme-linked immunosorbent assay | Homo sapiens | 1 | ALA3632527 | cell-based format | Scientific Literature | |
| 6. | ALA3636931 | A | Cytotoxicity against human T98G cells assessed as cell viability in the presence of PK11195 after 48 hrs by cell titer blue staining based fluorescence method | Homo sapiens | 5 | ALA3632527 | cell-based format | Scientific Literature | |
| 7. | ALA3636932 | A | Cytotoxicity against human T98G cells assessed as cell viability after 48 hrs by cell titer blue staining based fluorescence method | Homo sapiens | 5 | ALA3632527 | cell-based format | Scientific Literature | |
| 8. | ALA4699907 | B | Displacement of [3H]PK11195 from human TSPO A147T mutant expressed in HEK293 cells after 90 mins by scintillation counting method | Homo sapiens | 27 | ALA4699406 | cell-based format | Scientific Literature | |
| 9. | ALA4699908 | B | Displacement of [3H]PK11195 from wild-type human TSPO expressed in HEK293 cell membranes after 90 mins by scintillation counting method | Homo sapiens | 27 | ALA4699406 | cell membrane format | Scientific Literature | |
| 10. | ALA4699909 | B | Selectivity index, ratio of Ki for human TSPO A147T mutant expressed in HEK293 cell membranes to Ki for human TSPO expressed in HEK293 cell membranes | Homo sapiens | 27 | ALA4699406 | cell-based format | Scientific Literature |
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