| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3636666 | Binding | Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counter | Rattus norvegicus | 17 | ALA3632575 | cell-based format | Scientific Literature | |
| 2. | ALA3636667 | Binding | Displacement of [3H]diprenorphine from rat kappa-opioid receptor expressed in CHO cells after 90 mins by scintillation counter relative to zyklophin | Rattus norvegicus | 16 | ALA3632575 | cell-based format | Scientific Literature | |
| 3. | ALA3636668 | Binding | Displacement of [3H]DAMGO from rat mu-opioid receptor expressed in CHO cells after 90 mins by scintillation counter | Rattus norvegicus | 17 | ALA3632575 | cell-based format | Scientific Literature | |
| 4. | ALA3636669 | Binding | Selectivity ratio, ratio of Ki for rat mu-opioid receptor to Ki for rat kappa-opioid receptor | Rattus norvegicus | 17 | ALA3632575 | assay format | Scientific Literature | |
| 5. | ALA3636670 | Functional | Agonist activity at kappa-opioid receptor (unknown origin) at 10 uM after 90 mins by [35S]GTPgammaS binding assay | Homo sapiens | 14 | ALA3632575 | single protein format | Scientific Literature | |
| 6. | ALA3636673 | Functional | Antagonist activity at kappa-opioid receptor (unknown origin) assessed as inhibition of DynA(1-13)-induced [35S]-GTPgammaS binding after 90 mins | Homo sapiens | 5 | ALA3632575 | single protein format | Scientific Literature | |
| 7. | ALA3637218 | Functional | Antagonist activity at kappa-opioid receptor (unknown origin) assessed as inhibition of DynA(1-13)-induced [35S]-GTPgammaS binding after 90 mins relative to zyklophin | Homo sapiens | 1 | ALA3632575 | single protein format | Scientific Literature |
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