# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3705151 | B | Enzyme Assay: Enzyme assay using dipeptidyl peptidase-IV. | Homo sapiens | 8 | ALA3639302 | single protein format | BindingDB Database | |
2. | ALA3737789 | B | Inhibition of recombinant human DPP4 expressed in Sf9 cells using Gly-Pro-AMC substrate after 30 mins by plate reader analysis | Homo sapiens | 27 | ALA3734760 | cell-based format | Scientific Literature | |
3. | ALA3737790 | B | Inhibition of N-terminal FLAG tagged human QPP expressed in Sf9 cells using Nle-Pro-AMC substrate after 30 mins by plate reader analysis | Homo sapiens | 27 | ALA3734760 | cell-based format | Scientific Literature | |
4. | ALA3737791 | B | Inhibition of C-terminal His-tagged DPP8 (unknown origin) expressed in COS7 cells using H-Ala-Pro-pNA substrate preincubated for 15 mins | Homo sapiens | 27 | ALA3734760 | cell-based format | Scientific Literature | |
5. | ALA3737792 | B | Inhibition of bovine serum FAP | Bos taurus | 27 | ALA3734760 | single protein format | Scientific Literature | |
6. | ALA3737793 | A | Half life in rat at 1 mg/kg, iv and 2 mg/kg, po | Rattus norvegicus | 12 | ALA3734760 | organism-based format | Scientific Literature | |
7. | ALA3738361 | A | Plasma clearance in rat at 1 mg/kg, iv and 2 mg/kg, po | Rattus norvegicus | 12 | ALA3734760 | organism-based format | Scientific Literature | |
8. | ALA3738363 | A | Dose normalized AUC in rat at 1 mg/kg, iv and 2 mg/kg, po | Rattus norvegicus | 12 | ALA3734760 | organism-based format | Scientific Literature | |
9. | ALA3738364 | A | Oral bioavailability in rat at 2 mg/kg | Rattus norvegicus | 12 | ALA3734760 | organism-based format | Scientific Literature | |
10. | ALA3738370 | B | Selectivity index, ratio of IC50 for N-terminal FLAG tagged human QPP to IC50 for recombinant human DPP4 | Homo sapiens | 14 | ALA3734760 | assay format | Scientific Literature | |
11. | ALA3738371 | B | Selectivity index, ratio of IC50 for C-terminal His-tagged DPP8 (unknown origin) to IC50 for recombinant human DPP4 | Homo sapiens | 14 | ALA3734760 | assay format | Scientific Literature | |
12. | ALA3738372 | B | Selectivity index, ratio of IC50 for bovine serum FAP to IC50 for recombinant human DPP4 | 14 | ALA3734760 | assay format | Scientific Literature | ||
13. | ALA5247172 | B | Inhibition of DPP-4 (unknown origin) | Homo sapiens | 87 | ALA5244277 | single protein format | Scientific Literature |