# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3721241 | F | Inhibition of lipolysis in Sprague-Dawley rat epididymal adipocytes pre-incubated for 10 mins before theophylline addition followed by further incubation for 3 hrs by microplate reader based assay | Rattus norvegicus | 1 | cell-based format | Patent Bioactivity Data | ||
2. | ALA3721242 | F | Reduction in circulating free fatty acids in food-deprived Sprague-Dawley rat at 1 to 100 mg/kg, po measured after 10 to 240 mins post dose by NEFA assay | Rattus norvegicus | 1 | organism-based format | Patent Bioactivity Data | ||
3. | ALA3721243 | F | Reduction in circulating free fatty acids in food-deprived C57/B16 mouse at 100 mg/kg, ip measured after 30 mins by NEFA assay | Mus musculus | 3 | organism-based format | Patent Bioactivity Data | ||
4. | ALA3721244 | F | Agonist activity at human GPR81 expressed in CHO-K1 cell membranes pre-incubated for 5 to 10 mins before [35S]GTPgammaS addition followed by further incubation for 60 mins by microbeta counting based [35S]GTPgammaS binding assay | Homo sapiens | 142 | cell-based format | Patent Bioactivity Data | ||
5. | ALA3721245 | F | Agonist activity at human GPR81 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr by HTRF assay | Homo sapiens | 142 | cell-based format | Patent Bioactivity Data |