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# Aladdin ID Assay Type Description Organism Compounds Reference BAO Format Source 1. ALA3738314 Functional Agonist activity at TGR5 (unknown origin) assessed as cAMP level Homo sapiens 1 ALA3734669 single protein format Scientific Literature 2. ALA3738315 Binding Activation of human recombinant PXR up to 10 uM by alphascreen method Homo sapiens 2 ALA3734669 single protein format Scientific Literature 3. ALA3738317 ADME Cmax in mouse at 30 mg/kg, po administered as single dose by HPLC-MS analysis Mus musculus 2 ALA3734669 organism-based format Scientific Literature 4. ALA3738318 ADME AUC (0 to t) in mouse at 30 mg/kg, po administered as single dose by HPLC-MS analysis Mus musculus 2 ALA3734669 organism-based format Scientific Literature 5. ALA3738319 ADME Metabolic stability in mouse plasma assessed as compound remaining at 1 uM after 24 hrs by HPLC-ESI-MS/MS analysis Mus musculus 2 ALA3734669 cell-free format Scientific Literature 6. ALA3738320 Physicochemical n-octanol-water distribution coefficient, log D of the compound at pH 7.4 after 4 hrs by shake-flask method 2 ALA3734669 small-molecule physicochemical format Scientific Literature 7. ALA3738321 ADME Metabolic stability in mouse liver S9 fractions assessed as compound remaining at 1 uM after 1 hr by HPLC-ESI-MS/MS analysis in presence of NADPH regenerating system Mus musculus 2 ALA3734669 subcellular format Scientific Literature 8. ALA3738322 Physicochemical Kinetic solubility of the compound in NaCl solution at 25 deg C after 2 hrs by HPLC-ESI-MS/MS analysis 2 ALA3734669 small-molecule physicochemical format Scientific Literature 9. ALA4003652 ADME Drug metabolism in mouse liver microsomes assessed as (S)-3-((S)-4-((5R,8R,9S,10S,13R,14S,17R)-10,13-dimethyl-3-oxohexadecahydro-1H-cyclopenta[a]phenanthren-17-yl)pentanamido)-4-(1H-indol-3-yl)butanoic acid formation by HPLC-ESI-MS/MS analysis Mus musculus 1 ALA4002595 assay format Scientific Literature 10. ALA4003653 Binding Displacement of biotinylated ephrin-A1-Fc from recombinant mouse EphA2 receptor preincubated for 1 hr followed by biotinylated ephrin-A1-Fc addition measured after 4 hrs by ELISA method Mus musculus 17 ALA4002595 single protein format Scientific Literature 11. ALA4003655 Physicochemical n-Octanol-buffer partition co-efficient, log D of the compound at pH 7.4 incubated overnight by shake-flask method 3 ALA4002595 small-molecule physicochemical format Scientific Literature 12. ALA4003656 Physicochemical Kinetic solubility in MOPS buffer at pH 7.4 measured after 4 hrs by HPLC-ESI-MS/MS analysis 3 ALA4002595 small-molecule physicochemical format Scientific Literature 13. ALA4003657 ADME Stability in mouse plasma assessed as compound remaining at 1 uM after 24 hrs by HPLC-ESI-MS/MS analysis Mus musculus 3 ALA4002595 cell-free format Scientific Literature 14. ALA4003658 ADME Half-life in mouse liver microsomes at 1 uM in presence of NADPH by HPLC-ESI-MS/MS analysis Mus musculus 3 ALA4002595 assay format Scientific Literature 15. ALA4003659 ADME Cmax in mouse at 30 mg/kg, administered as single dose via oral gavage by HPLC-ESI-MS/MS analysis Mus musculus 3 ALA4002595 organism-based format Scientific Literature 16. ALA4003663 ADME Drug uptake in mouse plasma at 30 mg/kg, administered as single dose via oral gavage after 120 hrs by HPLC-ESI-MS/MS analysis Mus musculus 1 ALA4002595 organism-based format Scientific Literature 17. ALA4271244 ADME Cmax in mouse at 30 mg/kg, po Mus musculus 1 ALA4270498 organism-based format Scientific Literature 18. ALA4271245 Physicochemical Kinetic solubility of the compound 1 ALA4270498 small-molecule physicochemical format Scientific Literature 19. ALA4684876 Binding Competitive inhibition of biotinylated ephrin-A1-Fc binding to EphA2 (unknown origin) Homo sapiens 3 ALA4680187 single protein format Scientific Literature