| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3742597 | Binding | Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residual activity at 10 uM measured every 30 to 60 seconds for 60 mins | Homo sapiens | 58 | ALA3739299 | single protein format | Scientific Literature | |
| 2. | ALA3742598 | Binding | Inhibition of human Rce1-mediated CaaX protease activity using ABZ-KSKTKC(farnesyl)QIIM and ABZ-KSKTKC(farnesyl)VIQI as substrate assessed as residual activity measured every 30 to 60 seconds for 60 mins | Homo sapiens | 58 | ALA3739299 | single protein format | Scientific Literature | |
| 3. | ALA3742599 | ADME | Cytotoxicity against human HCT116 cells assessed as cell death at 25 uM after 20 hrs by celltiter blue assay (Rvb = 0.4%) | Homo sapiens | 31 | ALA3739299 | cell-based format | Scientific Literature |
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