| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3744105 | F | Antagonist activity against human GPR40 expressed in HEK293s FLPIN cells assessed as elaidic acid stimulated IP1 release after 2 hrs by TR-FRET analysis | Homo sapiens | 47 | ALA3739339 | cell-based format | Scientific Literature | |
| 2. | ALA3744106 | P | Lipophilicity, log D of the compound at pH 7.4 | 47 | ALA3739339 | small-molecule physicochemical format | Scientific Literature | ||
| 3. | ALA3744107 | P | Solubility of compound | 4 | ALA3739339 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA3744108 | A | Intrinsic clearance in rat hepatocytes measured per 10'6 cells | Rattus norvegicus | 3 | ALA3739339 | cell-based format | Scientific Literature | |
| 5. | ALA3744109 | A | Intrinsic clearance in human liver microsomes measured per 10'6 cells | Homo sapiens | 3 | ALA3739339 | tissue-based format | Scientific Literature | |
| 6. | ALA3744110 | B | Inhibition of human ERG | Homo sapiens | 3 | ALA3739339 | single protein format | Scientific Literature | |
| 7. | ALA3744111 | B | Antagonist activity against rat GPR40 | Rattus norvegicus | 3 | ALA3739339 | single protein format | Scientific Literature | |
| 8. | ALA3744112 | A | Fraction unbound in rat plasma | Rattus norvegicus | 3 | ALA3739339 | cell-free format | Scientific Literature | |
| 9. | ALA3744113 | A | Fraction unbound in human plasma | Homo sapiens | 3 | ALA3739339 | cell-free format | Scientific Literature | |
| 10. | ALA3744114 | A | Clearance in rat | Rattus norvegicus | 3 | ALA3739339 | organism-based format | Scientific Literature | |
| 11. | ALA3744115 | A | Unbound clearance in rat | Rattus norvegicus | 3 | ALA3739339 | organism-based format | Scientific Literature | |
| 12. | ALA3744116 | A | Volume of distribution at steady state in rat | Rattus norvegicus | 3 | ALA3739339 | organism-based format | Scientific Literature | |
| 13. | ALA3744117 | A | Oral bioavailability in rat | Rattus norvegicus | 3 | ALA3739339 | organism-based format | Scientific Literature | |
| 14. | ALA3744118 | A | Oral absorption in rat | Rattus norvegicus | 3 | ALA3739339 | organism-based format | Scientific Literature | |
| 15. | ALA3744119 | B | Antagonist activity at GPR43 (unkown origin) | Homo sapiens | 1 | ALA3739339 | single protein format | Scientific Literature | |
| 16. | ALA3744120 | B | Antagonist activity against pig Sodium/potassium-transporting ATPase | Sus scrofa | 1 | ALA3739339 | assay format | Scientific Literature | |
| 17. | ALA3744121 | F | Inhibition of NEFA-driven plasma insulin level in male Zucker rat pretreated with beta3-agonist for 30 mins at 80 mg/kg measured 4 hrs post dosing by ELISA | Rattus norvegicus | 1 | ALA3739339 | organism-based format | Scientific Literature | |
| 18. | ALA3744122 | A | Effect on plasma insulin level in male Zucker rat at 80 mg/kg measured after 4 hrs by ELISA relative to vehicle control | Rattus norvegicus | 1 | ALA3739339 | organism-based format | Scientific Literature | |
| 19. | ALA3744123 | A | Effect on plasma NEFA level in male Zucker rat at 80 mg/kg measured 4 hrs by ELISA assay relative to vehicle control | Rattus norvegicus | 1 | ALA3739339 | organism-based format | Scientific Literature | |
| 20. | ALA3744124 | B | Antagonist activity against mouse GPR40 | Mus musculus | 1 | ALA3739339 | single protein format | Scientific Literature |
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