| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3757432 | Binding | Displacement of [3H]DPCPX from adenosine A1 receptor in Sprague-Dawley rat whole brain after 1 hr by scintillation counting | Rattus norvegicus | 10 | ALA3751667 | assay format | Scientific Literature | |
| 2. | ALA3757433 | Binding | Displacement of [3H]NECA from adenosine A2A receptor in Sprague-Dawley rat striatal membrane after 1 hr by scintillation counting | Rattus norvegicus | 10 | ALA3751667 | assay format | Scientific Literature | |
| 3. | ALA3757434 | Binding | Selectivity ratio of Ki for adenosine A2A receptor in Sprague-Dawley rat striatal membrane to Ki for adenosine A1 receptor in Sprague-Dawley rat whole brain | Rattus norvegicus | 9 | ALA3751667 | assay format | Scientific Literature | |
| 4. | ALA3757435 | Functional | Reversal of haloperidol-induced catalepsy in Sprague-Dawley rat at 0.4 to 2 mg/kg, ip after 60 mins relative to control | Rattus norvegicus | 2 | ALA3751667 | organism-based format | Scientific Literature | |
| 5. | ALA3757436 | Physicochemical | n-octanol-potassium phosphate buffer partition coefficient, log D of the compound at pH 7.4 by shake flask method | 1 | ALA3751667 | small-molecule physicochemical format | Scientific Literature | ||
| 6. | ALA3757618 | Physicochemical | Solubility of the compound at 4.5 mg after 24 hrs by HPLC analysis | 1 | ALA3751667 | small-molecule physicochemical format | Scientific Literature | ||
| 7. | ALA5126825 | Binding | Binding affinity to human adenosine A2A receptor measured by radioligand-based affinity assay | Homo sapiens | 17 | ALA5126505 | single protein format | Scientific Literature | |
| 8. | ALA5126853 | Binding | Binding affinity to human adenosine A1A receptor measured by radioligand-based affinity assay | Homo sapiens | 12 | ALA5126505 | single protein format | Scientific Literature |
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