| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3756051 | B | Inhibition of recombinant human p70S6K assessed as residual activity at 1 uM by radiometric assay in presence of [gamma-33P]-ATP relative to control | Homo sapiens | 1 | ALA3751668 | single protein format | Scientific Literature | |
| 2. | ALA3756052 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 1 | ALA3751668 | single protein format | Scientific Literature | |
| 3. | ALA3756053 | A | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 1 | ALA3751668 | single protein format | Scientific Literature | |
| 4. | ALA3756054 | A | Inhibition of CYP2C9 (unknown origin) | Homo sapiens | 1 | ALA3751668 | single protein format | Scientific Literature | |
| 5. | ALA3756055 | A | Inhibition of CYP2C19 (unknown origin) | Homo sapiens | 1 | ALA3751668 | single protein format | Scientific Literature | |
| 6. | ALA3756056 | A | Half life in human liver microsomes | Homo sapiens | 1 | ALA3751668 | tissue-based format | Scientific Literature | |
| 7. | ALA3756057 | A | Cytotoxicity against mouse BAF3 cells after 48 hrs by MTT assay | Mus musculus | 22 | ALA3751668 | cell-based format | Scientific Literature | |
| 8. | ALA3756058 | B | Inhibition of TEL-fused Ret V804M mutant (unknown origin) expressed in mouse BA/F3 cells assessed as cell growth inhibition after 48 hrs by MTT assay | Homo sapiens | 23 | ALA3751668 | cell-based format | Scientific Literature | |
| 9. | ALA3756059 | A | Inhibition of CYP1A2 (unknown origin) | Homo sapiens | 1 | ALA3751668 | single protein format | Scientific Literature | |
| 10. | ALA3756060 | A | Cytotoxicity against human Nthy-ori 3-1 cells after 10 days by MTT assay | Homo sapiens | 23 | ALA3751668 | cell-based format | Scientific Literature | |
| 11. | ALA3756061 | B | Inhibition of wild type TEL-fused RET (unknown origin) expressed in mouse BA/F3 cells assessed as cell growth inhibition after 48 hrs by MTT assay | Homo sapiens | 23 | ALA3751668 | cell-based format | Scientific Literature | |
| 12. | ALA3756062 | B | Inhibition of recombinant human p70S6K by radiometric assay in presence of [gamma-33P]-ATP | Homo sapiens | 1 | ALA3751668 | single protein format | Scientific Literature | |
| 13. | ALA3756063 | B | Inhibition of recombinant human FLT4 by radiometric assay in presence of [gamma-33P]-ATP | Homo sapiens | 1 | ALA3751668 | single protein format | Scientific Literature | |
| 14. | ALA3756064 | B | Inhibition of TEL-fused wild type Ret (unknown origin) phosphorylation at Y1062/Y905 expressed in mouse BAF3 cells at 0.01 to 10 uM after 1 hr by Western blot analysis | Homo sapiens | 3 | ALA3751668 | cell-based format | Scientific Literature | |
| 15. | ALA3756065 | B | Inhibition of recombinant human RSK1 by radiometric assay in presence of [gamma-33P]-ATP | Homo sapiens | 1 | ALA3751668 | single protein format | Scientific Literature | |
| 16. | ALA3756066 | B | Inhibition of autophosphorylation of RET C634W mutant at Y905 in human TT cells at 1 uM after 4 hrs by Western blot analysis | Homo sapiens | 3 | ALA3751668 | cell-based format | Scientific Literature | |
| 17. | ALA3756067 | B | Inhibition of human wild type RET by radiometric assay in presence of [gamma-33P]-ATP | Homo sapiens | 21 | ALA3751668 | single protein format | Scientific Literature | |
| 18. | ALA3756068 | B | Inhibition of human Ret V804M mutant by radiometric assay in presence of [gamma-33P]-ATP | Homo sapiens | 19 | ALA3751668 | single protein format | Scientific Literature | |
| 19. | ALA3756070 | B | Inhibition of RET C634W mutant in human TT cells assessed as cell growth inhibition after 10 days by MTT assay | Homo sapiens | 23 | ALA3751668 | cell-based format | Scientific Literature | |
| 20. | ALA3756071 | B | Inhibition of human ERG assessed as prolongation of QT-interval at 100 uM by patch-clamp assay | Homo sapiens | 1 | ALA3751668 | single protein format | Scientific Literature |
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