| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3762573 | B | Binding affinity at delta opioid receptor (unknown origin) | Homo sapiens | 15 | ALA3758122 | single protein format | Scientific Literature | |
| 2. | ALA3762577 | B | Binding affinity at mu opioid receptor (unknown origin) | Homo sapiens | 16 | ALA3758122 | single protein format | Scientific Literature | |
| 3. | ALA3762762 | F | Analgesic activity in sc dosed rat by tail flick test | Rattus norvegicus | 2 | ALA3758122 | organism-based format | Scientific Literature | |
| 4. | ALA3802780 | B | Antagonist activity at DOR in CD1 mouse vas deferens assessed as reduction in DPDPE-induced inhibition of EFS-evoked contractions incubated for 60 mins | Mus musculus | 2 | ALA3797063 | tissue-based format | Scientific Literature | |
| 5. | ALA3802781 | B | Displacement of [3H]-DPN from rat MOR expressed in EE-HEK293 cell membranes by liquid scintillation counting | Rattus norvegicus | 7 | ALA3797063 | cell-based format | Scientific Literature | |
| 6. | ALA3802782 | B | Displacement of [3H]-DPN from rat DOR expressed in EE-HEK293 cell membranes by liquid scintillation counting | Rattus norvegicus | 7 | ALA3797063 | cell-based format | Scientific Literature | |
| 7. | ALA3802783 | B | Displacement of [3H]-DPN from human KOR expressed in EE-HEK293 cell membranes by liquid scintillation counting | Homo sapiens | 7 | ALA3797063 | cell-based format | Scientific Literature | |
| 8. | ALA3802784 | B | Selectivity index, ratio of Ki for rat DOR to Ki for rat MOR | Rattus norvegicus | 7 | ALA3797063 | assay format | Scientific Literature | |
| 9. | ALA3802785 | B | Selectivity index, ratio of Ki for human KOR to Ki for rat MOR | 7 | ALA3797063 | assay format | Scientific Literature | ||
| 10. | ALA3802786 | B | Agonist activity at MOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of EFS-induced contractions incubated for 60 mins | Cavia porcellus | 4 | ALA3797063 | tissue-based format | Scientific Literature | |
| 11. | ALA3802787 | B | Agonist activity at DOR in CD1 mouse vas deferens assessed as inhibition of EFS-induced contractions incubated for 60 mins | Mus musculus | 4 | ALA3797063 | tissue-based format | Scientific Literature | |
| 12. | ALA3802788 | B | Antagonist activity at DOR in CD1 mouse vas deferens assessed as pEC50 for DPDPE-induced inhibition of EFS-evoked contractions at 1 uM incubated for 60 mins | Mus musculus | 2 | ALA3797063 | tissue-based format | Scientific Literature | |
| 13. | ALA4058229 | B | Displacement of [3H]-DAMGO from MOR in rat brain membranes by liquid scintillation counting analysis | Rattus norvegicus | 6 | ALA4052787 | cell membrane format | Scientific Literature | |
| 14. | ALA4058230 | B | Displacement of [3H]-DPDPE from DOR in rat brain membranes by liquid scintillation counting analysis | Rattus norvegicus | 6 | ALA4052787 | cell membrane format | Scientific Literature | |
| 15. | ALA4058231 | B | Displacement of [3H]-(+)-U69,593 from KOR in guinea pig brain membranes by liquid scintillation counting analysis | Cavia porcellus | 6 | ALA4052787 | cell membrane format | Scientific Literature | |
| 16. | ALA4058232 | B | Ratio of Ki for DOR in rat brain membranes to Ki for MOR in rat brain membranes | Rattus norvegicus | 5 | ALA4052787 | cell membrane format | Scientific Literature | |
| 17. | ALA4058233 | B | Ratio of Ki for KOR in guinea pig brain membranes to Ki for MOR in rat brain membranes | 5 | ALA4052787 | cell membrane format | Scientific Literature | ||
| 18. | ALA4058234 | B | Agonist activity at MOR/KOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of electrically induced contractions after 5 mins | Cavia porcellus | 5 | ALA4052787 | assay format | Scientific Literature | |
| 19. | ALA4058235 | B | Agonist activity at DOR in CD-1 mouse vasa deferentia assessed as inhibition of electrically induced contractions after 5 mins | Mus musculus | 5 | ALA4052787 | assay format | Scientific Literature | |
| 20. | ALA4058236 | B | Antagonist activity at MOR in Dunkin-Hartley guinea pig ileum assessed as inhibition of electrically induced contractions after 5 mins by measuring ratio of IC50 for test compounds in presence and absence of NLX | Cavia porcellus | 4 | ALA4052787 | assay format | Scientific Literature |
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