| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3767697 | B | Inhibition of porcine pancreatic lipase at 30 uM | Sus scrofa | 4 | ALA3763072 | single protein format | Scientific Literature | |
| 2. | ALA3767698 | B | Inhibition of full length human C-terminal HA-tagged DAGLalpha expressed in HEK293 cells using DAG as substrate assessed as reduction in intracellular 2-AG level incubated for 20 mins by LC-MS analysis | Homo sapiens | 7 | ALA3763072 | cell-based format | Scientific Literature | |
| 3. | ALA3768666 | B | Inhibition of full length human C-terminal HA-tagged DAGLalpha expressed in HEK293 cell membrane using DAG as substrate incubated for 20 mins by LC-MS analysis | Homo sapiens | 31 | ALA3763072 | cell-based format | Scientific Literature | |
| 4. | ALA3768672 | B | Inhibition of MAGL (unknown origin) at 30 uM | Homo sapiens | 5 | ALA3763072 | single protein format | Scientific Literature | |
| 5. | ALA3768871 | A | Permeability coefficient of compound at pH 5.5 after 4 hrs by PAMPA | 10 | ALA3763072 | assay format | Scientific Literature | ||
| 6. | ALA3768873 | B | Ratio of IC50 for full length human C-terminal HA-tagged DAGLalpha expressed in HEK293 cells assessed as reduction in intracellular 2-AG level to IC50 for full length human C-terminal HA-tagged DAGLalpha expressed in HEK293 cell membrane | Homo sapiens | 6 | ALA3763072 | cell-based format | Scientific Literature | |
| 7. | ALA3768874 | B | Inhibition of DAGLbeta (unknown origin) | Homo sapiens | 6 | ALA3763072 | single protein format | Scientific Literature | |
| 8. | ALA3768875 | B | Selectivity ratio of IC50 for full length human C-terminal HA-tagged DAGLalpha expressed in HEK293 cell membrane to IC50 for DAGLbeta (unknown origin) | Homo sapiens | 4 | ALA3763072 | cell-based format | Scientific Literature |
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