| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3768207 | B | Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysis | Rattus norvegicus | 28 | assay format | Scientific Literature | ||
| 2. | ALA3768208 | B | Antagonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assay | Homo sapiens | 28 | cell-based format | Scientific Literature | ||
| 3. | ALA3768209 | B | Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D2 receptor after 45 mins by microplate scintillation counting analysis | Rattus norvegicus | 28 | assay format | Scientific Literature | ||
| 4. | ALA3768210 | B | Displacement of [3H]-dofetilide from human ERG potassium channel by scintillation proximity assay | Homo sapiens | 28 | single protein format | Scientific Literature | ||
| 5. | ALA3768215 | A | Inhibition of human CYP1A2 expressed in bactosome | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 6. | ALA3768216 | A | Inhibition of human CYP2C9 expressed in bactosome | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 7. | ALA3768217 | A | Inhibition of human CYP2C19 expressed in bactosome | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 8. | ALA3768218 | A | Inhibition of human CYP2D6 expressed in bactosome | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 9. | ALA3768219 | A | Inhibition of human CYP3A4 expressed in bactosome using DBOMF as substrate | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 10. | ALA3768220 | A | Inhibition of human CYP3A4 expressed in bactosome using 7BQ as substrate | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 11. | ALA3768221 | A | Intrinsic clearance in human liver microsomes assessed per mg of protein | Homo sapiens | 4 | tissue-based format | Scientific Literature | ||
| 12. | ALA3768222 | A | Intrinsic clearance in rat liver microsomes assessed per mg of protein | Rattus norvegicus | 3 | tissue-based format | Scientific Literature | ||
| 13. | ALA3768229 | A | Fraction unbound in portal vein-cannulated rat blood | Rattus norvegicus | 4 | tissue-based format | Scientific Literature | ||
| 14. | ALA3768230 | A | Fraction unbound in portal vein-cannulated rat brain | Rattus norvegicus | 4 | tissue-based format | Scientific Literature | ||
| 15. | ALA3768231 | B | Agonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assay | Homo sapiens | 28 | cell-based format | Scientific Literature | ||
| 16. | ALA3768232 | B | Selectivity ratio of Ki for rat brain dopamine D2 receptor to Ki for rat brain dopamine D3 receptor | Rattus norvegicus | 5 | assay format | Scientific Literature | ||
| 17. | ALA3768418 | B | Selectivity ratio of Ki for rat brain dopamine D2 receptor to Ki for human ERG | 4 | assay format | Scientific Literature |
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