# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3772516 | B | Inhibition of human recombinant KLK4 expressed in Escherichia coli using Bachem I-1120 as substrate preincubated for 15 mins followed by substrate addition by microplate reader analysis | Homo sapiens | 11 | ALA3769401 | assay format | Scientific Literature | |
2. | ALA3772517 | B | Inhibition of human recombinant KLK2 expressed in Escherichia coli using Bachem I-1295 as substrate preincubated for 15 mins followed by substrate addition by microplate reader analysis | Homo sapiens | 11 | ALA3769401 | assay format | Scientific Literature | |
3. | ALA3772518 | B | Inhibition of human recombinant KLK1 expressed in Escherichia coli using Bachem I-1295 as substrate preincubated for 15 mins followed by substrate addition by microplate reader analysis | Homo sapiens | 11 | ALA3769401 | assay format | Scientific Literature | |
4. | ALA3772679 | B | Inhibition of human recombinant KLK8 expressed in Escherichia coli using Bachem I-1120 as substrate preincubated for 15 mins followed by substrate addition by microplate reader analysis | Homo sapiens | 11 | ALA3769401 | assay format | Scientific Literature | |
5. | ALA3772680 | B | Inhibition of recombinant uPA (unknown origin) using Biophen CS-61(44) as substrate | Homo sapiens | 11 | ALA3769401 | single protein format | Scientific Literature | |
6. | ALA3772681 | B | Inhibition of recombinant tPA (unknown origin) using Biophen CS-05(88) as substrate | Homo sapiens | 11 | ALA3769401 | single protein format | Scientific Literature | |
7. | ALA3772682 | B | Inhibition of human plasma thrombin using Biophen CS-21(66) as substrate preincubated for 15 mins followed by substrate addition by microplate reader analysis | Homo sapiens | 11 | ALA3769401 | cell-free format | Scientific Literature | |
8. | ALA3772683 | B | Inhibition of human plasma plasmin using Biophen CS-21(66) as substrate | Homo sapiens | 10 | ALA3769401 | cell-free format | Scientific Literature | |
9. | ALA3772684 | B | Inhibition of factor 10a (unknown origin) using Biophen CS-11(32) as substrate | Homo sapiens | 11 | ALA3769401 | single protein format | Scientific Literature | |
10. | ALA3772685 | B | Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate by 5-5'-Dithiobis(2 nitrobenzoic acid)-based assay | Electrophorus electricus | 10 | ALA3769401 | single protein format | Scientific Literature | |
11. | ALA3772687 | B | Irreversible inhibition of human recombinant KLK2 expressed in Escherichia coli using H-Pro-Phe-Arg-AMC as fluorogenic substrate at 100 times IC50 preincubated for 15 mins followed by 100 fold dilution measured for 1 hr | Homo sapiens | 2 | ALA3769401 | assay format | Scientific Literature | |
12. | ALA3772690 | B | Reversible inhibition of human recombinant KLK8 expressed in Escherichia coli using Boc-Val-Pro-Arg-AMC as fluorogenic substrate at 100 times IC50 preincubated for 15 mins followed by 100 fold dilution measured for 1 hr | Homo sapiens | 3 | ALA3769401 | assay format | Scientific Literature | |
13. | ALA3772692 | B | Reversible inhibition of recombinant uPA (unknown origin) using Biophen CS-61(44) as substrate at 100 times IC50 preincubated for 15 mins followed by 100 fold dilution measured for 1 hr | Homo sapiens | 1 | ALA3769401 | single protein format | Scientific Literature | |
14. | ALA3772706 | B | Reversible inhibition of human recombinant KLK4 expressed in Escherichia coli using Bachem I-1120 as fluorogenic substrate at 100 times IC50 preincubated for 15 mins followed by 100 fold dilution measured for 1 hr by microplate reader analysis | Homo sapiens | 7 | ALA3769401 | assay format | Scientific Literature |