| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3772523 | ADME | Apparent permeability across apical to basolateral side in MDCK cells at 10 uM after 60 mins | Canis lupus familiaris | 14 | ALA3769359 | cell-based format | Scientific Literature | |
| 2. | ALA3772524 | Binding | Inhibition of human ERG at 10 uM by patch clamp assay | Homo sapiens | 14 | ALA3769359 | assay format | Scientific Literature | |
| 3. | ALA3772525 | Binding | Inhibition of human recombinant PAK1 kinase domain using coumarin/fluorescein-labeled FRET peptide as substrate preincubated for 10 mins followed by ATP addition measured after 60 mins by Z-LYTE assay | Homo sapiens | 14 | ALA3769359 | single protein format | Scientific Literature | |
| 4. | ALA3772526 | Binding | Inhibition of PAK1 in human EBC1 cells assessed as reduction in levels of MEK phosphorylation at S298 residue after 2 hrs by HTRF assay | Homo sapiens | 14 | ALA3769359 | cell-based format | Scientific Literature | |
| 5. | ALA3772527 | ADME | Hepatic clearance in human liver microsomes after 1 hr by LC-MS/MS analysis | Homo sapiens | 8 | ALA3769359 | tissue-based format | Scientific Literature |
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