| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3779310 | B | Inhibition of recombinant human His-tagged TRIM24-PHD/bromodomain expressed in Escherichia coli strains BL21 (DE3) cells using biotinylated H3K23ac (1 to 33 residues) peptide after 1 hr by AlphaScreen assay | Homo sapiens | 38 | ALA3774340 | cell-based format | Scientific Literature | |
| 2. | ALA3779311 | B | Inhibition of recombinant human BAZ2A expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 3. | ALA3779312 | B | Inhibition of recombinant human ATAD2B expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 4. | ALA3779313 | B | Inhibition of recombinant human ATAD2A expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 5. | ALA3779314 | B | Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay | Homo sapiens | 23 | ALA3774340 | cell-based format | Scientific Literature | |
| 6. | ALA3779315 | P | Kinetic solubility of compound in phosphate buffer at pH 7 | 16 | ALA3774340 | small-molecule physicochemical format | Scientific Literature | ||
| 7. | ALA3779317 | B | Ratio of EC50 for Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells to IC50 for recombinant human His-tagged TRIM24-PHD/bromodomain expressed in Escherichia coli strains BL21 (DE3) cells | Homo sapiens | 13 | ALA3774340 | cell-based format | Scientific Literature | |
| 8. | ALA3779318 | B | Binding affinity to recombinant human His-tagged TRIM24-PHD/bromodomain expressed in Escherichia coli strains BL21 (DE3) cells by isothermal titration calorimetry | Homo sapiens | 1 | ALA3774340 | cell-based format | Scientific Literature | |
| 9. | ALA3779319 | B | Binding affinity to BRPF1 (unknown origin) expressed in Escherichia coli strains BL21 (DE3) cells by isothermal titration calorimetry | Homo sapiens | 1 | ALA3774340 | cell-based format | Scientific Literature | |
| 10. | ALA3779320 | B | Binding affinity to recombinant human TRIM24-PHD/bromodomain expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 11. | ALA3779321 | B | Binding affinity to recombinant human BRPF1 expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 12. | ALA3779322 | B | Binding affinity to recombinant human BRPF2 expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 13. | ALA3779323 | B | Binding affinity to recombinant human BRPF3 expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 14. | ALA3779324 | B | Binding affinity to recombinant human BAZ2B expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 15. | ALA3779325 | B | Binding affinity to recombinant human TAF1 bromodomain 2 expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 16. | ALA3776805 | B | Binding affinity to recombinant human BRD4 long isoform bromodomain 1 expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 17. | ALA3776806 | B | Binding affinity to recombinant human BRD4 long isoform bromodomain 2 expressed in bacterial system by bromoscan assay | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 18. | ALA3776807 | B | Inhibition of recombinant human BRD2 isoform 1 bromodomain 2 expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 19. | ALA3777024 | B | Inhibition of recombinant human BRD3 bromodomain 1 expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature | |
| 20. | ALA3777025 | B | Inhibition of recombinant human BRD3 bromodomain 2 expressed in bacterial system assessed as residual activity at 1 uM by bromoscan assay relative to control | Homo sapiens | 1 | ALA3774340 | assay format | Scientific Literature |
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