# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3778805 | B | Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for 10 mins measured after 20 mins by alphascreen assay | Homo sapiens | 56 | ALA3774338 | assay format | Scientific Literature | |
2. | ALA3778806 | B | Inhibition of recombinant human N-terminal GST-tagged KDM4B (1 to 500 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 as substrate preincubated for 10 mins measured after 20 mins by alphascreen assay | Homo sapiens | 56 | ALA3774338 | cell-based format | Scientific Literature | |
3. | ALA3778807 | B | Inhibition of KDM5B (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins by alphascreen assay | Homo sapiens | 56 | ALA3774338 | single protein format | Scientific Literature | |
4. | ALA3778979 | B | Inhibition of KDM5C (unknown origin) using biotin-H3K4me3 as substrate preincubated for 15 mins followed by substrate addition measured after 20 mins by alphascreen assay | Homo sapiens | 54 | ALA3774338 | single protein format | Scientific Literature | |
5. | ALA3776392 | B | Inhibition of KDM2A (unknown origin) using biotin-H3K36me2 (28 to 48 residues) as substrate at 100 uM preincubated for 15 mins followed by substrate addition measured after 30 mins by alphascreen assay relative to control | Homo sapiens | 2 | ALA3774338 | single protein format | Scientific Literature | |
6. | ALA3776393 | B | Inhibition of KDM6B (unknown origin) using biotin-H3K27me3 (21 to 44 residues) as substrate at 100 uM preincubated for 15 mins followed by substrate addition measured after 5 mins by alphascreen assay relative to control | Homo sapiens | 5 | ALA3774338 | single protein format | Scientific Literature |