| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3778163 | B | Inhibition of human KDM6B catalytic domain using H3(20 to 36 residues)K27Me3 peptide as substrate assessed as demethylation of substrate by Rapidfire mass spectrometric analysis | Homo sapiens | 18 | ALA3774367 | single protein format | Scientific Literature | |
| 2. | ALA3778164 | B | Inhibition of KDM4C (unknown origin) using H3K9Me3 peptide as substrate assessed as demethylation of substrate by Rapidfire mass spectrometric analysis | Homo sapiens | 34 | ALA3774367 | single protein format | Scientific Literature | |
| 3. | ALA3778166 | B | Inhibition of full length His-MBP-att-EGLN3 (1 to 239 residues) (unknown origin) in Escherichia coli BL21(DE3)pRR692 cells assessed as hydroxylation of the cy-5 labelled C-terminal oxygen dependent domain of substrate Hif2A preincubated for 30 mins followed by substrate addition measured after 40 mins by TR-FRET assay | Homo sapiens | 10 | ALA3774367 | assay format | Scientific Literature | |
| 4. | ALA3778167 | B | Selectivity ratio of IC50 for human KDM6B catalytic domain to IC50 for KDM4C (unknown origin) | Homo sapiens | 6 | ALA3774367 | assay format | Scientific Literature |
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