| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3776820 | B | Inhibition of human RORgamma ligand binding domain (Serine 253 to Lysine 518 residues) expressed in CHOK1 cells incubated for 2 days by Gal4 luciferase reporter gene assay | Homo sapiens | 28 | cell-based format | Scientific Literature | ||
| 2. | ALA3776821 | B | Inhibition of mouse RORgamma ligand binding domain (Isoleucine 251 to Lysine 516) expressed in CHOK1 cells incubated for 2 days by Gal4 luciferase reporter gene assay | Mus musculus | 28 | cell-based format | Scientific Literature | ||
| 3. | ALA3776822 | A | Metabolic stability in liver S9 fraction (unknown origin) assessed as parent compound remaining incubated for 10 mins | Homo sapiens | 14 | subcellular format | Scientific Literature | ||
| 4. | ALA3776823 | A | Metabolic stability in liver S9 fraction (unknown origin) assessed as parent compound remaining incubated for 60 mins | Homo sapiens | 14 | subcellular format | Scientific Literature | ||
| 5. | ALA3776824 | A | Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate preincubated with substrate for 5 mins followed by NADPH addition measured after 20 mins by HPLC analysis | Homo sapiens | 3 | tissue-based format | Scientific Literature | ||
| 6. | ALA3776825 | B | Inhibition of human GST-tagged RORgamma ligand binding domain (253 to 518 residues) expressed in sf9 cells using biotin-EEPSLLKKLLLAPA by FRET assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 7. | ALA3776833 | A | Inhibition of CYP2C9 in human liver microsomes using diclofenac as substrate preincubated with substrate for 5 mins followed by NADPH addition measured after 20 mins by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 8. | ALA3776834 | A | Inhibition of CYP2D6 in human liver microsomes using bufuralol as substrate preincubated with substrate for 5 mins followed by NADPH addition measured after 20 mins by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 9. | ALA3776835 | A | Inhibition of CYP1A2 in human liver microsomes using ethoxyresorufin as substrate preincubated with substrate for 5 mins followed by NADPH addition measured after 20 mins by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 10. | ALA3776836 | A | Inhibition of CYP2A6 in human liver microsomes using coumarin as substrate preincubated with substrate for 5 mins followed by NADPH addition measured after 20 mins by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 11. | ALA3776837 | A | Inhibition of CYP2C19 in human liver microsomes using S-mephenytoin as substrate preincubated with substrate for 5 mins followed by NADPH addition measured after 20 mins by HPLC analysis | Homo sapiens | 1 | tissue-based format | Scientific Literature | ||
| 12. | ALA3776838 | B | Inhibition of human RORalpha | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA3776839 | B | Inhibition of human SF-1 receptor | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA3776840 | B | Inhibition of human RORbeta | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA3776841 | B | Inhibition of mouse GR | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 16. | ALA3776842 | B | Inhibition of human RXRalpha | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA3776843 | B | Inhibition of human VDR | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA3776844 | B | Inhibition of human FXR | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA3776845 | B | Inhibition of mouse LXRalpha | Mus musculus | 1 | single protein format | Scientific Literature | ||
| 20. | ALA3778098 | B | Inhibition of human PPARalpha | Homo sapiens | 1 | single protein format | Scientific Literature |
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