| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3778013 | B | Inhibition of human factor 9a using CH3SO2-DCHG-Gly-Arg-AFC.AcOH as substrate preinubated for 30 mins followed by substrate addition measured after 1 hr by fluorescence assay | Homo sapiens | 5 | ALA3774356 | single protein format | Scientific Literature | |
| 2. | ALA3778020 | B | Competitive binding affinity to human factor 9a expressed in Escherichia coli after 30 mins by ALIS-AS analysis in presence of (S)-2,6-Dichloro-N-(2-(7-fluoro-2-methyl-1H-benzo[d]-imidazol-5-yl)2-(3-fluorophenyl)ethyl)-4-(3-methyl-1H-1,2,4-triazol-1-yl)benzamide | Homo sapiens | 4 | ALA3774356 | assay format | Scientific Literature | |
| 3. | ALA3778021 | A | Drug level in human liver microsomes treated with (R)-2,6-Dichloro-N-(2-(3-fluorophenyl)-2-(2-methyl-1Hbenzo[d]imidazol-5-yl)ethyl)-4-(3-methyl-1H-1,2,4-triazol-1-yl)-benzamide after 4 hrs by LC-MS/MS analysis | Homo sapiens | 4 | ALA3774356 | tissue-based format | Scientific Literature | |
| 4. | ALA3778025 | A | Drug level in Sprague-Dawley rat liver microsomes treated with (R)-2,6-Dichloro-N-(2-(3-fluorophenyl)-2-(2-methyl-1Hbenzo[d]imidazol-5-yl)ethyl)-4-(3-methyl-1H-1,2,4-triazol-1-yl)-benzamide after 4 hrs by LC-MS/MS analysis | Rattus norvegicus | 4 | ALA3774356 | tissue-based format | Scientific Literature | |
| 5. | ALA3778028 | A | Drug level in beagle dog liver microsomes treated with (R)-2,6-Dichloro-N-(2-(3-fluorophenyl)-2-(2-methyl-1Hbenzo[d]imidazol-5-yl)ethyl)-4-(3-methyl-1H-1,2,4-triazol-1-yl)-benzamide at 100 uM after 4 hrs by LC-MS/MS analysis | Canis lupus familiaris | 4 | ALA3774356 | tissue-based format | Scientific Literature | |
| 6. | ALA3778030 | P | Retention time of the compound by size exclusion chromatography | 4 | ALA3774356 | small-molecule physicochemical format | Scientific Literature |
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