| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3783739 | B | Inhibition of matripase/hepsin/hepatocyte growth factor activator-mediated HGF activation in human 18Co fibroblasts assessed as scattering of human DU145 cells after 24 hrs by crystal violet staining method | Homo sapiens | 4 | ALA3779883 | cell-based format | Scientific Literature | |
| 2. | ALA3783740 | P | Kinetic solubility of the compound at pH 7.4 | 7 | ALA3779883 | small-molecule physicochemical format | Scientific Literature | ||
| 3. | ALA3783741 | P | Lipophilicity, logD of the compound at pH 7.4 by shake-flask method | 7 | ALA3779883 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA3783753 | B | Selectivity ratio of Ki for human recombinant factor 10a to Ki for human recombinant hepsin | Homo sapiens | 2 | ALA3779883 | assay format | Scientific Literature | |
| 5. | ALA3783755 | B | Selectivity ratio of Ki for human recombinant factor 10a to Ki for human recombinant matripase | Homo sapiens | 1 | ALA3779883 | assay format | Scientific Literature | |
| 6. | ALA3782550 | B | Inhibition of human recombinant matripase catalytic domain using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysis | Homo sapiens | 19 | ALA3779883 | single protein format | Scientific Literature | |
| 7. | ALA3782551 | B | Inhibition of human recombinant hepsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysis | Homo sapiens | 19 | ALA3779883 | single protein format | Scientific Literature | |
| 8. | ALA3782552 | B | Inhibition of human recombinant hepatocyte growth factor activator using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysis | Homo sapiens | 19 | ALA3779883 | cell-based format | Scientific Literature | |
| 9. | ALA3782553 | B | Inhibition of human recombinant trypsin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysis | Homo sapiens | 19 | ALA3779883 | protein format | Scientific Literature | |
| 10. | ALA3782596 | B | Inhibition of human recombinant thrombin using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysis | Homo sapiens | 19 | ALA3779883 | single protein format | Scientific Literature | |
| 11. | ALA3782597 | B | Inhibition of human recombinant factor 10a using H2N(EEdansyl)GKQLRVVNGG (KDabcyl)-NH2 as substrate by fluorometric analysis | Homo sapiens | 19 | ALA3779883 | single protein format | Scientific Literature |
The page will load shortly, Thanks for your patience!