| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3789169 | B | Inhibition of KDM4E (unknown origin) preincubated for 15 mins followed by histone substrate addition measured after 1 hr by alphascreen assay | Homo sapiens | 1 | ALA3784917 | single protein format | Scientific Literature | |
| 2. | ALA3791433 | B | Inhibition of KDM2A (unknown origin) preincubated for 15 mins followed by histone substrate addition measured after 1 hr by alphascreen assay | Homo sapiens | 1 | ALA3784917 | single protein format | Scientific Literature | |
| 3. | ALA3791434 | B | Inhibition of KDM3A (unknown origin) preincubated for 15 mins followed by histone substrate addition measured after 1 hr by alphascreen assay | Homo sapiens | 1 | ALA3784917 | single protein format | Scientific Literature | |
| 4. | ALA3791435 | B | Inhibition of KDM5C (unknown origin) preincubated for 15 mins followed by histone substrate addition measured after 1 hr by alphascreen assay | Homo sapiens | 1 | ALA3784917 | single protein format | Scientific Literature | |
| 5. | ALA3791436 | B | Inhibition of KDM6B (unknown origin) preincubated for 15 mins followed by histone substrate addition measured after 1 hr by alphascreen assay | Homo sapiens | 1 | ALA3784917 | single protein format | Scientific Literature | |
| 6. | ALA3791437 | B | Inhibition of KDM4C (unknown origin) preincubated for 15 mins followed by histone substrate addition measured after 1 hr by alphascreen assay | Homo sapiens | 1 | ALA3784917 | single protein format | Scientific Literature | |
| 7. | ALA3791438 | B | Inhibition of PHD2 (unknown origin) preincubated for 15 mins followed by histone substrate addition measured after 1 hr by alphascreen assay | Homo sapiens | 1 | ALA3784917 | single protein format | Scientific Literature | |
| 8. | ALA3791439 | B | Inhibition of FIH (unknown origin) using ankyrin peptide substrate preincubated for 5 mins followed by substrate addition measured after 5 mins MALDI-TOF mass spectrometric analysis | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature | |
| 9. | ALA3791440 | B | Inhibition of full-length FLAG-tagged KDM4A (unknown origin) expressed in human HeLa cells assessed as increase in H3K9me3 level after 24 hrs by DAPI staining based immunofuorescence assay | Homo sapiens | 1 | ALA3784917 | cell-based format | Scientific Literature | |
| 10. | ALA3791441 | B | Inhibition of KDM4A in human MCF7 cells assessed as increase in H3K9me3 level after 24 hrs by DAPI staining based immunofuorescence assay | Homo sapiens | 1 | ALA3784917 | cell-based format | Scientific Literature | |
| 11. | ALA3791446 | B | Selectivity ratio of IC50 for KDM3A (unknown origin) to IC50 for KDM4C (unknown origin) | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature | |
| 12. | ALA3791447 | B | Selectivity ratio of IC50 for KDM5C (unknown origin) to IC50 for KDM4C (unknown origin) | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature | |
| 13. | ALA3791448 | B | Selectivity ratio of IC50 for KDM6B (unknown origin) to IC50 for KDM4C (unknown origin) | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature | |
| 14. | ALA3791449 | B | Selectivity ratio of IC50 for PHD2 (unknown origin) to IC50 for KDM4C (unknown origin) | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature | |
| 15. | ALA3791450 | B | Selectivity ratio of IC50 for FIH (unknown origin) to IC50 for KDM4C (unknown origin) | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature | |
| 16. | ALA3791451 | B | Selectivity ratio of IC50 for KDM3A (unknown origin) to IC50 for KDM4E (unknown origin) | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature | |
| 17. | ALA3791452 | B | Selectivity ratio of IC50 for KDM5C (unknown origin) to IC50 for KDM4E (unknown origin) | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature | |
| 18. | ALA3791453 | B | Selectivity ratio of IC50 for KDM6B (unknown origin) to IC50 for KDM4E (unknown origin) | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature | |
| 19. | ALA3791454 | B | Selectivity ratio of IC50 for PHD2 (unknown origin) to IC50 for KDM4E (unknown origin) | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature | |
| 20. | ALA3791455 | B | Selectivity ratio of IC50 for FIH (unknown origin) to IC50 for KDM4E (unknown origin) | Homo sapiens | 1 | ALA3784917 | assay format | Scientific Literature |
The page will load shortly, Thanks for your patience!