| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3791458 | Binding | Competitive inhibition of recombinant His6-tagged KDM2A (1 to 517 residues) (unknown origin) expressed in Escherichia coli BL21 cells using methylstat as substrate preincubated for 30 mins followed by substrate addition measured after 4 hrs by fluorescence polarization assay | Homo sapiens | 3 | ALA3784917 | cell-based format | Scientific Literature | |
| 2. | ALA3791701 | Binding | Competitive inhibition of recombinant His6-tagged KDM4A (1 to 359 residues) (unknown origin) expressed in Escherichia coli BL21 cells using methylstat as substrate preincubated for 30 mins followed by substrate addition measured after 4 hrs by fluorescence polarization assay | Homo sapiens | 3 | ALA3784917 | cell-based format | Scientific Literature | |
| 3. | ALA3791702 | Binding | Inhibition of KDM2A in human MIAPaCa2 cells assessed as increase in H3K36me2 level after 48 hrs by Hoechst 33258 staining based immunofluorescence assay | Homo sapiens | 3 | ALA3784917 | cell-based format | Scientific Literature | |
| 4. | ALA3791703 | Binding | Inhibition of KDM2A in human MIAPaCa2 cells assessed as increase in H3K9me3 level after 48 hrs by Hoechst 33258 staining based immunofluorescence assay | Homo sapiens | 3 | ALA3784917 | cell-based format | Scientific Literature | |
| 5. | ALA3791704 | Functional | Growth inhibition of human MIAPaCa2 cells after 48 hrs by CellTiter-Glo assay | Homo sapiens | 3 | ALA3784917 | cell-based format | Scientific Literature |
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