| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3788932 | B | Inhibition of recombinant human C-terminal FLAG-tagged KDM5A (1 to 1090 residues) expressed in baculovirus infected sf9 cells using biotin-H3K4me3 substrate incubated for 30 mins by TR-FRET assay | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 2. | ALA3788933 | B | Inhibition of recombinant human N-terminal His-FLAG-tagged KDM5B (2 to 751 residues) expressed in baculovirus infected sf9 cells using biotin-H3K4me3 substrate incubated for 30 mins by TR-FRET assay | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 3. | ALA3788934 | B | Inhibition of recombinant human N-terminal GST-tagged KDM4C (2 to 372 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 substrate incubated for 30 mins by TR-FRET assay | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
| 4. | ALA3788936 | B | Inhibition of recombinant human C-terminal FLAG-tagged KDM2B (1 to 650 residues) expressed in baculovirus infected sf9 cells using biotin-H3K36me2 substrate incubated for 30 mins by alphascreen assay | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 5. | ALA3788937 | B | Inhibition of KDM5A in human ZR-75-1 cells assessed as reduction in H3K4me3 demethylation incubated for 72 hrs by fluorometric immunoassay | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 6. | ALA3788938 | B | Inhibition of KDM5B in human ZR-75-1 cells assessed as reduction in H3K4me3 demethylation incubated for 72 hrs by fluorometric immunoassay | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 7. | ALA4223290 | B | Inhibition of KDM5A (unknown origin) preincubated with enzyme | Homo sapiens | 23 | single protein format | Scientific Literature | ||
| 8. | ALA4223291 | B | Inhibition of KDM5B (unknown origin) preincubated with enzyme | Homo sapiens | 34 | single protein format | Scientific Literature | ||
| 9. | ALA4223292 | B | Inhibition of KDM4C (unknown origin) preincubated with enzyme | Homo sapiens | 29 | single protein format | Scientific Literature | ||
| 10. | ALA4223293 | B | Inhibition of KDM5A/KDM5B in human ZR-75-1 cells assessed as increase in H3K4me3 level after 72 hrs by fluorometric immunoassay | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 11. | ALA4223294 | B | Inhibition of KDM5A/KDM5B in human ZR-75-1 cells assessed as increase in H3K4me3 level after 72 hrs by fluorometric immunoassay relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA4223295 | B | Inhibition of KDM1A (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4223296 | B | Inhibition of KDM2A (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA4223297 | B | Inhibition of KDM2B (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA4223298 | B | Inhibition of KDM3A (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA4223299 | B | Inhibition of KDM4A (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA4223300 | B | Inhibition of KDM4B (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA4223301 | B | Inhibition of KDM4D (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA4223302 | B | Inhibition of KDM4E (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA4223303 | B | Inhibition of KDM6B (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature |
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