| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3788932 | B | Inhibition of recombinant human C-terminal FLAG-tagged KDM5A (1 to 1090 residues) expressed in baculovirus infected sf9 cells using biotin-H3K4me3 substrate incubated for 30 mins by TR-FRET assay | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 2. | ALA3788933 | B | Inhibition of recombinant human N-terminal His-FLAG-tagged KDM5B (2 to 751 residues) expressed in baculovirus infected sf9 cells using biotin-H3K4me3 substrate incubated for 30 mins by TR-FRET assay | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 3. | ALA3788934 | B | Inhibition of recombinant human N-terminal GST-tagged KDM4C (2 to 372 residues) expressed in baculovirus infected sf9 cells using biotin-H3K9me3 substrate incubated for 30 mins by TR-FRET assay | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
| 4. | ALA3788935 | B | Inhibition of recombinant human N-terminal His-tagged KDM4A (1 to 350 residues) expressed in Escherichia coli using biotin-H3K9me3 substrate incubated for 30 mins by TR-FRET assay | Homo sapiens | 5 | assay format | Scientific Literature | ||
| 5. | ALA3789194 | B | Selectivity ratio of IC50 for recombinant human C-terminal FLAG-tagged KDM5A (1 to 1090 residues) expressed in baculovirus infected sf9 cells to IC50 for recombinant human N-terminal GST-tagged KDM4C (2 to 372 residues) expressed in baculovirus infected sf9 cells | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 6. | ALA3789195 | B | Selectivity ratio of IC50 for recombinant human N-terminal His-FLAG-tagged KDM5B (2 to 751 residues) expressed in baculovirus infected sf9 cells to IC50 for recombinant human N-terminal GST-tagged KDM4C (2 to 372 residues) expressed in baculovirus infected sf9 cells | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 7. | ALA3789196 | B | Selectivity ratio of IC50 for recombinant human N-terminal His-tagged KDM4A (1 to 350 residues) expressed in Escherichia coli to IC50 for recombinant human N-terminal GST-tagged KDM4C (2 to 372 residues) expressed in baculovirus infected sf9 cells | Homo sapiens | 3 | cell-based format | Scientific Literature |
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