| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3794750 | B | Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using fluorescence labelled srctide as substrate by mobility shift assay in presence of ATP | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 2. | ALA3794752 | B | Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using 5-FAM-peptide 2 as substrate after 2 hrs by electrophoretic mobility shift assay in presence of ATP | Homo sapiens | 27 | ALA3792292 | assay format | Scientific Literature | |
| 3. | ALA3794761 | B | Inhibition of full length human N-terminal His-tagged ABL (2 to 1130 residues) expressed in baculovirus expression system using fluorescence labelled ABLtide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 4. | ALA3794762 | B | Inhibition of full length human N-terminal GST-tagged CSK (1 to 450 residues) expressed in baculovirus expression system using fluorescence labelled srctide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 5. | ALA3794763 | B | Inhibition of human N-terminal GST-tagged EGFR cytoplasmic domain (669 to 1210 residues) expressed in baculovirus expression system using fluorescence labelled srctide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 6. | ALA3794764 | B | Inhibition of human N-terminal GST-tagged EPHA2 cytoplasmic domain (572 to 976 residues) expressed in baculovirus expression system using fluorescence labelled Blk/Lyntide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 7. | ALA3794765 | B | Inhibition of human N-terminal GST-tagged EPHB4 cytoplasmic domain (577 to 987 residues) expressed in baculovirus expression system using fluorescence labelled Blk/Lyntide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 8. | ALA3794766 | B | Inhibition of human N-terminal GST-tagged FGFR1 cytoplasmic domain (398 to 822 residues) expressed in baculovirus expression system using fluorescence labelled CSKtide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 9. | ALA3794767 | B | Inhibition of human N-terminal GST-tagged FLT3 cytoplasmic domain (564 to 993 residues) expressed in baculovirus expression system using fluorescence labelled srctide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 10. | ALA3794768 | B | Inhibition of human N-terminal GST-tagged IGF1R cytoplasmic domain (959 to 1367 residues) expressed in baculovirus expression system using fluorescence labelled IRS1 as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 11. | ALA3794769 | B | Inhibition of full length human N-terminal GST-tagged ITK (2 to 620 residues) expressed in baculovirus expression system using fluorescence labelled srctide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 12. | ALA3794770 | B | Inhibition of human N-terminal His-tagged JAK3 catalytic domain (795 to 1124 residues) expressed in baculovirus expression system using fluorescence labelled srctide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 13. | ALA3794771 | B | Inhibition of human N-terminal GST-tagged KDR cytoplasmic domain (790 to 1356 residues) expressed in baculovirus expression system using fluorescence labelled CSKtide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 14. | ALA3794772 | B | Inhibition of full length human N-terminal GST-tagged LCK (1 to 500 residues) expressed in baculovirus expression system using fluorescence labelled srctide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 15. | ALA3794773 | B | Inhibition of human N-terminal GST-tagged MET cytoplasmic domain (956 to 1390 residues) expressed in baculovirus expression system using fluorescence labelled srctide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 16. | ALA3794774 | B | Inhibition of human N-terminal GST-tagged PDGFRalpha cytoplasmic domain (550 to 1089 residues) expressed in baculovirus expression system using fluorescence labelled CSKtide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 17. | ALA3794818 | B | Inhibition of full length human N-terminal GST-tagged PYK2 (1 to 967 residues) expressed in baculovirus expression system using fluorescence labelled Blk/Lyntide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 18. | ALA3794819 | B | Inhibition of full length human N-terminal GST-tagged SRC (1 to 536 residues) expressed in baculovirus expression system using fluorescence labelled srctide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 19. | ALA3794820 | B | Inhibition of full length human N-terminal GST-tagged SYK (1 to 635 residues) expressed in baculovirus expression system using fluorescence labelled Blk/Lyntide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature | |
| 20. | ALA3794821 | B | Inhibition of human N-terminal GST-tagged TIE2 receptor cytoplasmic domain (771 to 1124 residues) expressed in baculovirus expression system using fluorescence labelled Blk/Lyntide as substrate at 50 times IC50 by electrophoretic mobility shift assay relative to control | Homo sapiens | 3 | ALA3792292 | assay format | Scientific Literature |
The page will load shortly, Thanks for your patience!