| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3796231 | B | Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by substrate addition measured after 1 hr by spectrofluorimetric analysis | Homo sapiens | 45 | ALA3792352 | single protein format | Scientific Literature | |
| 2. | ALA3796232 | F | Cytotoxicity against human RPMI8226 cells assessed as cell viability after 72 hrs by CellTiter 96 aqueous one solution cell proliferation assay | Homo sapiens | 3 | ALA3792352 | cell-based format | Scientific Literature | |
| 3. | ALA3796233 | F | Cytotoxicity against human ARH77 cells assessed as cell viability after 72 hrs by CellTiter 96 aqueous one solution cell proliferation assay | Homo sapiens | 3 | ALA3792352 | cell-based format | Scientific Literature | |
| 4. | ALA3796234 | F | Cytotoxicity against human U266B1 cells assessed as cell viability after 72 hrs by CellTiter 96 aqueous one solution cell proliferation assay | Homo sapiens | 3 | ALA3792352 | cell-based format | Scientific Literature | |
| 5. | ALA3796235 | A | Elimination half life in Sprague-Dawley rat at 1 mg/kg, caudal iv by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 6. | ALA3796236 | A | Elimination half life in Sprague-Dawley rat at 0.2 mg/kg, ig through feeding tube by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 7. | ALA3796237 | A | Tmax in Sprague-Dawley rat at 1 mg/kg, caudal iv by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 8. | ALA3796238 | A | Tmax in Sprague-Dawley rat at 0.2 mg/kg, ig through feeding tube by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 9. | ALA3796239 | A | Cmax in Sprague-Dawley rat at 1 mg/kg, caudal iv by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 10. | ALA3796240 | A | Cmax in Sprague-Dawley rat at 0.2 mg/kg, ig through feeding tube by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 11. | ALA3796241 | A | AUClast in Sprague-Dawley rat at 1 mg/kg, caudal iv by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 12. | ALA3796242 | A | AUClast in Sprague-Dawley rat at 0.2 mg/kg, ig through feeding tube by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 13. | ALA3796243 | A | AUC(0 to infinity) in Sprague-Dawley rat at 1 mg/kg, caudal iv by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 14. | ALA3796244 | A | AUC(0 to infinity) in Sprague-Dawley rat at 0.2 mg/kg, ig through feeding tube by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 15. | ALA3796245 | A | MRTlast in Sprague-Dawley rat at 1 mg/kg, caudal iv by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 16. | ALA3796246 | A | MRTlast in Sprague-Dawley rat at 0.2 mg/kg, ig through feeding tube by LC/MS/MS analysis | Rattus norvegicus | 1 | ALA3792352 | organism-based format | Scientific Literature | |
| 17. | ALA3796247 | F | Cell cycle arrest in human U266 cells assessed as accumulation at S phase at 10 nM by propidium iodide/RNase staining based flow cytometric analysis (Rvb = 29.47 %) | Homo sapiens | 1 | ALA3792352 | cell-based format | Scientific Literature | |
| 18. | ALA3796248 | F | Cell cycle arrest in human U266 cells assessed as accumulation at G1 phase at 10 nM by propidium iodide/RNase staining based flow cytometric analysis (Rvb = 58.21 %) | Homo sapiens | 1 | ALA3792352 | cell-based format | Scientific Literature | |
| 19. | ALA3796249 | F | Cell cycle arrest in human U266 cells assessed as accumulation at G2/M phase at 10 nM by propidium iodide/RNase staining based flow cytometric analysis (Rvb = 12.33 %) | Homo sapiens | 1 | ALA3792352 | cell-based format | Scientific Literature |
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