| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3804623 | B | Inhibition of recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity expressed in Escherichia coli BL21-Codonplus (DE3)-RIL cells using MTOB as substrate after 15 mins by NADH consumption assay | Homo sapiens | 25 | ALA3797021 | cell-based format | Scientific Literature | |
| 2. | ALA3804624 | F | Cytotoxicity against human HCT116 p53-/- cells assessed as inhibition of cell growth after 72 hrs by MTT assay | Homo sapiens | 15 | ALA3797021 | cell-based format | Scientific Literature | |
| 3. | ALA3804625 | B | Inhibition of rabbit muscle L-lactate dehydrogenase using sodium pyruvate as substrate measured every 10 secs for 30 mins by microplate reader method | Oryctolagus cuniculus | 4 | ALA3797021 | assay format | Scientific Literature | |
| 4. | ALA3804626 | B | Selectivity ratio of IC50 for rabbit muscle L-lactate dehydrogenase to IC50 for recombinant His6-tagged CtBP2 (31 to 384 residues) (unknown origin) dehydrogenase activity | 3 | ALA3797021 | assay format | Scientific Literature | ||
| 5. | ALA3804627 | P | Aqueous stability in pH 7.2 phosphate buffer at 4 mM after 72 hrs by HPLC method | 3 | ALA3797021 | small-molecule physicochemical format | Scientific Literature | ||
| 6. | ALA3804628 | B | Inhibition of CtBP2 (unknown origin) transfected in human HCT116 p53-/- cells assessed as increase in Bik transcription at 2 mM by dual luciferase reporter gene assay relative to control | Homo sapiens | 6 | ALA3797021 | cell-based format | Scientific Literature | |
| 7. | ALA3804629 | B | Inhibition of CtBP2 (unknown origin) transfected in human HCT116 p53-/- cells assessed as increase in Bik transcription at 4 mM by dual luciferase reporter gene assay relative to control | Homo sapiens | 3 | ALA3797021 | cell-based format | Scientific Literature |
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