| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3803236 | B | Inhibition of human recombinant N-terminal GST-tagged LRRK2 (968 residues) expressed in baculovirus infected sf9 cells using LRRKtide as substrate at 100 uM incubated for 10 mins by scintillation counting method in presence of [gamma33P]ATP | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 2. | ALA3803238 | B | Inhibition of human recombinant GST-tagged LRRK2 G2019S mutant (970 residues) expressed in baculovirus expression system using LRRKtide as substrate at 100 uM incubated for 10 mins by scintillation counting method in presence of [gamma33P]ATP | Homo sapiens | 6 | assay format | Scientific Literature | ||
| 3. | ALA3803240 | B | Inhibition of human recombinant N-terminal GST-tagged LRRK2 (968 residues) expressed in baculovirus infected sf9 cells using LRRKtide as substrate incubated for 10 mins by scintillation counting method in presence of [gamma33P]ATP | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 4. | ALA3803241 | B | Inhibition of human recombinant GST-tagged LRRK2 G2019S mutant (970 residues) expressed in baculovirus expression system using LRRKtide as substrate incubated for 10 mins by scintillation counting method in presence of [gamma33P]ATP | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 5. | ALA3803242 | B | Selectivity ratio of ID50 for human recombinant N-terminal GST-tagged LRRK2 (968 residues) expressed in baculovirus infected sf9 cells to ID50 for human recombinant GST-tagged LRRK2 G2019S mutant (970 residues) expressed in baculovirus expression system | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 6. | ALA3803243 | B | Inhibition of full length human recombinant N-terminal His6-tagged SRC expressed in baculovirus infected sf21 cells using KVEKIGEGTYGVVYK as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 7. | ALA3803244 | B | Inhibition of full length human recombinant N-terminal GST-tagged GSK3beta expressed in baculovirus infected sf9 cells using GSK3 substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 8. | ALA3803245 | B | Inhibition of full length human recombinant N-terminal GST-His6-tagged HCK (M1 to P505 residues) expressed in baculovirus infected sf9 cells using KVEKIGEGTYGVVYK as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 9. | ALA3803246 | B | Inhibition of human recombinant FAK expressed in baculovirus infected sf9 cells using KVEKIGEGTYGVVYK as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 10. | ALA3803247 | B | Inhibition of full length human recombinant N-terminal His-tagged CDK6/N-terminal GST-tagged Cyclin D1 expressed in baculovirus infected sf9 cells using RB-CTF as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 11. | ALA3803248 | B | Inhibition of recombinant rat N-terminal GST-tagged DYRK1A (1 to 499 residues) expressed in Escherichia coli using KKISGRLSPIMTEQ-NH2 as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Rattus norvegicus | 4 | assay format | Scientific Literature | ||
| 12. | ALA3801083 | B | Inhibition of human recombinant N-terminal His-tagged ABL (27 residues) expressed in baculovirus infected sf9 cells using KKGEAIYAAPFA-NH2 as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 13. | ALA3801084 | B | Inhibition of human recombinant N-terminal GST-His6-tagged FLT3 (R571-S993 residues) expressed in baculovirus infected sf9 cells using KVEKIGEGTYGVVYK as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 14. | ALA3801085 | B | Inhibition of full length human recombinant N-terminal GST-tagged CDK2 (M1-L298 residues)/Cyclin A2 (M1-L432 residues) expressed in baculovirus infected sf9 cells using histone H1 as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 15. | ALA3801086 | B | Inhibition of full length human recombinant N-terminal GST-His6-tagged CDK9 (M1-F372 residues)/Cyclin T1 (M1-K726 residues) expressed in baculovirus infected sf9 cells using CDKtide as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 16. | ALA3801087 | B | Inhibition of full length human recombinant N-terminal GST-tagged CDK9/Cyclin K expressed in baculovirus infected sf9 cells using CDKtide as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 17. | ALA3801088 | B | Inhibition of full length human recombinant N-terminal GST-tagged CDK4/Cyclin D1 expressed in baculovirus infected sf9 cells using RB-CTF as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 18. | ALA3801089 | B | Inhibition of full length human recombinant N-terminal GST-His-tagged PI4KB expressed in sf9 cells using phosphatidyl inositol:phosphatidyl serine (1:3) substrate at 100 uM by ADP-Glo kinase assay relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 19. | ALA3801090 | B | Inhibition of full length human recombinant N-terminal GST-tagged PIM1 expressed in Escherichia coli using S6 Kinase/Rsk2 peptide2 as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 20. | ALA3801091 | B | Competitive inhibition of human recombinant GST-tagged LRRK2 G2019S mutant (970 residues) expressed in baculovirus expression system assessed as enzyme-inhibitor complex by Michaelis-Menten kinetics in presence of varying level of ATP | Homo sapiens | 1 | assay format | Scientific Literature |
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