Inhibition of human PDGFRalpha using (poly [Glu, Tyr] 4:1) as substrate assessed as incorporation of 33P in substrate by [gamma33P] ATP-based kinase assay
Inhibition of PI3Kalpha (unknown origin) using (poly [Glu, Tyr] 4:1) as substrate assessed as incorporation of 33P in substrate by [gamma33P] ATP-based kinase assay
Inhibition of PI3Kbeta (unknown origin) using (poly [Glu, Tyr] 4:1) as substrate assessed as incorporation of 33P in substrate by [gamma33P] ATP-based kinase assay
Inhibition of PI3Kgamma (unknown origin) using (poly [Glu, Tyr] 4:1) as substrate assessed as incorporation of 33P in substrate by [gamma33P] ATP-based kinase assay
Inhibition of PI3Kdelta (unknown origin) using (poly [Glu, Tyr] 4:1) as substrate assessed as incorporation of 33P in substrate by [gamma33P] ATP-based kinase assay
Antiproliferative activity against human U87 cells assessed as reduction in cell viability at 3 to 300 uM incubated for 5 days by Prestoblue reagent based assay
Antiproliferative activity against human T98 cells assessed as reduction in cell viability at 3 to 300 uM incubated for 5 days by Prestoblue reagent based assay