| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3802845 | Binding | Inhibition of N-terminal FLAG-tagged ERK1 (unknown origin) expressed in baculovirus preincubated for 5 mins using myelin basic protein as substrate measured after 60 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 2. | ALA3802846 | Binding | Inhibition of C-terminal 6His-tagged CDK2/N-terminal GST-tagged cyclin A (unknown origin) expressed in baculovirus preincubated for 5 mins using histone-H1 as substrate measured after 20 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 3. | ALA3802847 | Binding | Inhibition of N-terminal FLAG-tagged p38alpha (unknown origin) expressed in baculovirus preincubated for 5 mins using myelin basic protein as substrate measured after 60 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 4. | ALA3802848 | Binding | Inhibition of full length human CDC7 co-expressed with N-terminal GST-tagged ASK in baculovirus preincubated for 5 mins using MCM2 as substrate measured after 60 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA3797131 | single protein format | Scientific Literature | |
| 5. | ALA3802849 | Binding | Inhibition of N-terminal FLAG-tagged PLK1 (unknown origin) expressed in baculovirus preincubated for 5 mins using alpha-casein as substrate measured after 60 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 6. | ALA3802850 | Binding | Inhibition of N-terminal 6His-tagged PI3Kalpha (unknown origin) co-expressed with p85alpha in baculovirus using L-alpha-phosphatidyl-D-myo-inositol 4,5-diphosphate as substrate measured after 60 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA3797131 | single protein format | Scientific Literature | |
| 7. | ALA3802851 | Binding | Inhibition of ROCK2 (unknown origin) | Homo sapiens | 1 | ALA3797131 | single protein format | Scientific Literature | |
| 8. | ALA3802852 | Binding | Inhibition of N-terminal FLAG-tagged PKCzeta (unknown origin) expressed in baculovirus preincubated for 5 mins using fluorescein-PKC substrate measured after 60 mins in presence of ATP by TR-FRET assay | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 9. | ALA3802853 | Binding | Inhibition of N-terminal His6-tagged recombinant human c-Met preincubated for 5 mins measured after 10 mins in presence of ATP by AlphaScreen assay | Homo sapiens | 1 | ALA3797131 | single protein format | Scientific Literature | |
| 10. | ALA3802854 | Binding | Inhibition of full length N-terminal His-tagged recombinant human SRC preincubated for 5 mins measured after 10 mins in presence of ATP by AlphaScreen assay | Homo sapiens | 1 | ALA3797131 | single protein format | Scientific Literature | |
| 11. | ALA3802855 | Binding | Inhibition of N-terminal FLAG-tagged FAK cytoplasmic domain (unknown origin) expressed in baculovirus preincubated for 5 mins measured after 20 mins in presence of ATP by AlphaScreen assay | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 12. | ALA3802856 | Binding | Inhibition of N-terminal FLAG-tagged PKCalpha (unknown origin) expressed in baculovirus preincubated for 5 mins using fluorescein-PKC substrate measured after 60 mins in presence of ATP by TR-FRET assay | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 13. | ALA3802857 | Binding | Inhibition of N-terminal FLAG-tagged PKCbeta (unknown origin) expressed in baculovirus preincubated for 5 mins using fluorescein-PKC substrate measured after 60 mins in presence of ATP by TR-FRET assay | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 14. | ALA3802858 | Binding | Inhibition of N-terminal FLAG-tagged PKCdelta (unknown origin) expressed in baculovirus preincubated for 5 mins using fluorescein-PKC substrate measured after 60 mins in presence of ATP by TR-FRET assay | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 15. | ALA3802859 | Binding | Inhibition of CLK (unknown origin) | Homo sapiens | 1 | ALA3797131 | single protein format | Scientific Literature | |
| 16. | ALA3802860 | Binding | Inhibition of N-terminal GST-tagged GSK-3beta (unknown origin) expressed in baculovirus preincubated for 5 mins using GSK3 substrate peptide measured after 60 mins in presence of [gamma-33P]ATP by scintillation counting method | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 17. | ALA3802861 | Binding | Inhibition of N-terminal GST-tagged human TrkA expressed in baculovirus preincubated for 5 mins measured after 10 mins in presence of ATP by AlphaScreen assay | Homo sapiens | 1 | ALA3797131 | assay format | Scientific Literature | |
| 18. | ALA3802862 | Functional | Inhibition of T-activator CD3/CD28 stimulated IL2 production in human whole blood measured after 24 hrs by ELISA | Homo sapiens | 1 | ALA3797131 | tissue-based format | Scientific Literature | |
| 19. | ALA3802863 | Functional | Inhibition of anti-CD3-antibody-induced IL2 production in Balb/c mouse administered orally as single dose followed anti-CD3 challenge measured after 1 hr by ELISA | Mus musculus | 1 | ALA3797131 | organism-based format | Scientific Literature | |
| 20. | ALA3802864 | ADME | Plasma concentration in Balb/c mouse at 10 mg/kg to 100 mg/kg, po after 4 hrs | Mus musculus | 1 | ALA3797131 | organism-based format | Scientific Literature |
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