| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3802887 | Binding | Inhibition of PI3Kalpha mutant in human BT474 cells assessed as inhibition of AKT phosphorylation at Thr-308 residue after 2 hrs by ELISA | Homo sapiens | 17 | ALA3797054 | cell-based format | Scientific Literature | |
| 2. | ALA3802888 | Binding | Inhibition of PI3Kbeta in PTEN deficient human MDA-MB-468 cells assessed as inhibition of AKT phosphorylation at Ser-473 residue after 2 hrs by plate reader analysis | Homo sapiens | 17 | ALA3797054 | cell-based format | Scientific Literature | |
| 3. | ALA3802890 | Physicochemical | Lipophilicity, log D of compound at pH 7.4 | 16 | ALA3797054 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA3802891 | ADME | Intrinsic clearance in human hepatocytes assessed per million cells | Homo sapiens | 15 | ALA3797054 | cell-based format | Scientific Literature | |
| 5. | ALA3802892 | Physicochemical | Solubility in pH 7.4 phosphate buffer using solid compound | 12 | ALA3797054 | small-molecule physicochemical format | Scientific Literature | ||
| 6. | ALA3802893 | ADME | Apparent permeability from apical to basolateral side in human Caco2 cells at 10 uM for 2 hrs by LC-MS/MS analysis | Homo sapiens | 11 | ALA3797054 | cell-based format | Scientific Literature | |
| 7. | ALA3802894 | ADME | AUC in hairy mouse at 30 umol/kg, po | Mus musculus | 8 | ALA3797054 | organism-based format | Scientific Literature |
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