| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3807033 | B | Inhibition of His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo assay in presence of MgATP | Homo sapiens | 25 | ALA3804808 | assay format | Scientific Literature | |
| 2. | ALA3807034 | B | Inhibition of His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) using glucose as substrate after 45 mins by ADP-glo assay in presence of MgATP | Homo sapiens | 25 | ALA3804808 | assay format | Scientific Literature | |
| 3. | ALA3807035 | B | Selectivity ratio of IC50 for His-tagged human HK1 (11 to 917 residues) expressed in Escherichia coli BL21(DE3) to IC50 for His-tagged human HK2 (17 to 916 residues) expressed in Escherichia coli BL21(DE3) | Homo sapiens | 2 | ALA3804808 | assay format | Scientific Literature | |
| 4. | ALA3807036 | B | Inhibition of HK2 in human UM-UC-3 cells using 2FDG as substrate assessed as suppression of G6P production preincubated for 30 mins followed by substrate treatment for 90 mins by resazurin assay | Homo sapiens | 3 | ALA3804808 | cell-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!