| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3811360 | B | Inhibition of full length C-terminal hexahistidine tagged GRK2 (unknown origin) S670A mutant expressed in High Five cells using Bac to Bac insect cell expression system using tubulin as substrate by SDS-PAGE method | Homo sapiens | 27 | ALA3808388 | cell-based format | Scientific Literature | |
| 2. | ALA3811361 | B | Inhibition of GRK1 (unknown origin) using tubulin as substrate by SDS-PAGE method | Homo sapiens | 27 | ALA3808388 | single protein format | Scientific Literature | |
| 3. | ALA3811362 | B | Inhibition of GRK5 (unknown origin) using tubulin as substrate by SDS-PAGE method | Homo sapiens | 27 | ALA3808388 | single protein format | Scientific Literature | |
| 4. | ALA3811363 | B | Inhibition of PKA (unknown origin) using CREBtide as substrate by ADP-Glo kinase assay | Homo sapiens | 27 | ALA3808388 | assay format | Scientific Literature | |
| 5. | ALA3811364 | B | Inhibition of ROCK1 (unknown origin) at 10 uM by ADP-Glo kinase assay | Homo sapiens | 4 | ALA3808388 | single protein format | Scientific Literature | |
| 6. | ALA3811367 | B | Selectivity ratio of IC50 for GRK5 (unknown origin) to IC50 for full length C-terminal hexahistidine tagged GRK2 (unknown origin) S670A mutant expressed in High Five cells using the Bac to Bac insect cell expression system | Homo sapiens | 7 | ALA3808388 | cell-based format | Scientific Literature | |
| 7. | ALA3811373 | B | Inhibition of GRK2 in C57BL/6 mouse cardiomyocytes assessed as increase in contractility at 0.5 uM preincubated for 10 mins followed by beta adrenergic receptor agonist isoproterenol addition for 2 mins | Mus musculus | 3 | ALA3808388 | cell-based format | Scientific Literature | |
| 8. | ALA4043633 | B | Inhibition of GRK2 (unknown origin) | Homo sapiens | 5 | ALA4043080 | single protein format | Scientific Literature | |
| 9. | ALA4043634 | B | Inhibition of bovine GRK2 S670A mutant after 5 mins in presence of ATP by phosphorimaging assay | Bos taurus | 34 | ALA4043080 | assay format | Scientific Literature | |
| 10. | ALA4043635 | B | Inhibition of bovine GRK1 (1 to 535 residues) after 5 mins after 5 mins in presence of ATP by phosphorimaging assay | Bos taurus | 34 | ALA4043080 | single protein format | Scientific Literature | |
| 11. | ALA4043636 | B | Inhibition of bovine GRK5 after 5 mins after 5 mins in presence of ATP by phosphorimaging assay | Bos taurus | 34 | ALA4043080 | single protein format | Scientific Literature | |
| 12. | ALA4043637 | B | Inhibition of mouse PKA using CREBtide as substrate after 30 mins in presence of ATP by ADP-Glo kinase assay | Mus musculus | 34 | ALA4043080 | assay format | Scientific Literature | |
| 13. | ALA4043638 | B | Inhibition of ROCK1 (unknown origin) at 10 uM by ADP-Glo kinase assay | Homo sapiens | 34 | ALA4043080 | single protein format | Scientific Literature | |
| 14. | ALA4043643 | A | Half life in CD-1 mouse liver microsomes at 1 uM measured up to 60 mins in presence of NADPH by LC-MS/MS analysis | Mus musculus | 13 | ALA4043080 | assay format | Scientific Literature |
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