| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3812305 | B | Inhibition of human wild type partial length CSF1R expressed in bacterial expression system assessed as residual activity at 1 uM by KinomeScan method | Homo sapiens | 1 | ALA3808357 | assay format | Scientific Literature | |
| 2. | ALA3812306 | B | Inhibition of human wild type partial length DDR1 expressed in bacterial expression system assessed as residual activity at 1 uM by KinomeScan method | Homo sapiens | 1 | ALA3808357 | assay format | Scientific Literature | |
| 3. | ALA3812307 | B | Inhibition of human wild type partial length cKIT expressed in bacterial expression system assessed as residual activity at 1 uM by KinomeScan method | Homo sapiens | 1 | ALA3808357 | assay format | Scientific Literature | |
| 4. | ALA3812308 | B | Inhibition of human wild type partial length PDGFRbeta expressed in bacterial expression system assessed as residual activity at 1 uM by KinomeScan method | Homo sapiens | 1 | ALA3808357 | assay format | Scientific Literature | |
| 5. | ALA3812309 | B | Inhibition of His-tagged recombinant human CSF1R expressed in baculovirus expression system after 1 hr by Z-lyte assay | Homo sapiens | 1 | ALA3808357 | assay format | Scientific Literature | |
| 6. | ALA3812310 | B | Inhibition of GST-tagged human DDR1 expressed in baculovirus after 1 hr by Z-lyte assay | Homo sapiens | 1 | ALA3808357 | assay format | Scientific Literature | |
| 7. | ALA3812311 | B | Inhibition of N-terminal GST-tagged recombinant human PDGFRbeta (amino acids 557-end) expressed in baculovirus infected insect Sf9 cells using Poly(4:1 Glu, Tyr) peptide as substrate after 1 hr by promega ADP-glo assay | Homo sapiens | 1 | ALA3808357 | cell-based format | Scientific Literature | |
| 8. | ALA3812312 | B | Inhibition of His-tagged human recombinant cKIT expressed in baculovirus using Tyr 06 peptide as substrate after 1 hr by Z-lyte assay | Homo sapiens | 1 | ALA3808357 | assay format | Scientific Literature | |
| 9. | ALA3812313 | A | Antiproliferative activity against mouse BAF3 cells | Mus musculus | 29 | ALA3808357 | cell-based format | Scientific Literature | |
| 10. | ALA3812314 | B | Inhibition of Tel-fused cKIT (unknown origin) transfected in mouse BAF3 cells assessed as decrease in cell proliferation after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 29 | ALA3808357 | cell-based format | Scientific Literature | |
| 11. | ALA3812315 | B | Inhibition of Tel-fused cKIT V559D mutant (unknown origin) transfected in mouse BAF3 cells assessed as decrease in cell proliferation after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 3 | ALA3808357 | cell-based format | Scientific Literature | |
| 12. | ALA3812316 | B | Inhibition of Tel-fused cKIT V559D/V654A double mutant (unknown origin) transfected in mouse BAF3 cells assessed as decrease in cell proliferation after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 3 | ALA3808357 | cell-based format | Scientific Literature | |
| 13. | ALA3812317 | B | Inhibition of Tel-fused cKIT N822K mutant (unknown origin) transfected in mouse BAF3 cells assessed as decrease in cell proliferation after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 3 | ALA3808357 | cell-based format | Scientific Literature | |
| 14. | ALA3812318 | B | Inhibition of Tel-fused cKIT T670I mutant (unknown origin) transfected in mouse BAF3 cells assessed as decrease in cell proliferation after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 3 | ALA3808357 | cell-based format | Scientific Literature | |
| 15. | ALA3812319 | B | Inhibition of Tel-fused cKIT V654A mutant (unknown origin) transfected in mouse BAF3 cells assessed as decrease in cell proliferation after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 3 | ALA3808357 | cell-based format | Scientific Literature | |
| 16. | ALA3812320 | B | Inhibition of Tel-fused cKIT L567P mutant (unknown origin) transfected in mouse BAF3 cells assessed as decrease in cell proliferation after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 3 | ALA3808357 | cell-based format | Scientific Literature | |
| 17. | ALA3812497 | B | Inhibition of Tel-fused cKIT T670I/V559D double mutant (unknown origin) transfected in mouse BAF3 cells assessed as decrease in cell proliferation after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 3 | ALA3808357 | cell-based format | Scientific Literature | |
| 18. | ALA3812498 | B | Inhibition of Tel-fused cKIT D816V mutant (unknown origin) transfected in mouse BAF3 cells assessed as decrease in cell proliferation after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 3 | ALA3808357 | cell-based format | Scientific Literature | |
| 19. | ALA3812499 | F | Antiproliferative activity against cKIT dependent human GISTT1 cells assessed as reduction in cell viability after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 3 | ALA3808357 | cell-based format | Scientific Literature | |
| 20. | ALA3812500 | F | Antiproliferative activity against FLT3-ITD dependent human MV4-11 cells assessed as reduction in cell viability after 72 hrs by celltiter-glo/CCK8 assay | Homo sapiens | 3 | ALA3808357 | cell-based format | Scientific Literature |
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