# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3815552 | Functional | Cytotoxicity against human K562 cells after 72 hrs by MTT assay | Homo sapiens | 4 | ALA3813662 | cell-based format | Scientific Literature | |
2. | ALA3815553 | Functional | Cytotoxicity against human HCT116 cells after 72 hrs by MTT assay | Homo sapiens | 4 | ALA3813662 | cell-based format | Scientific Literature | |
3. | ALA3815554 | Binding | Inhibition of human full length (His)6-tagged PKCalpha expressed in insect Sf21 cells using histone H1 as substrate assessed as residual enzyme activity at 10 uM measured for 30 mins by [gamma-33P]ATP-based kinase assay | Homo sapiens | 4 | ALA3813662 | cell-based format | Scientific Literature | |
4. | ALA3815555 | Binding | Inhibition of human full length (His)6-tagged PKCalpha expressed in insect Sf21 cells using histone H1 as substrate assessed as residual enzyme activity at 1 uM measured for 30 mins by [gamma-33P]ATP-based kinase assay | Homo sapiens | 4 | ALA3813662 | cell-based format | Scientific Literature | |
5. | ALA3815556 | Binding | Inhibition of human full length (His)6-tagged PKCgamma expressed in insect Sf21 cells using histone H1 as substrate assessed as residual enzyme activity at 10 uM measured for 30 mins by [gamma-33P]ATP-based kinase assay | Homo sapiens | 4 | ALA3813662 | cell-based format | Scientific Literature | |
6. | ALA3815557 | Binding | Inhibition of human full length (His)6-tagged PKCgamma expressed in insect Sf21 cells using histone H1 as substrate assessed as residual enzyme activity at 1 uM measured for 30 mins by [gamma-33P]ATP-based kinase assay | Homo sapiens | 4 | ALA3813662 | cell-based format | Scientific Literature | |
7. | ALA3815558 | Binding | Inhibition of human full length (His)6-tagged Pim-1 expressed in insect Sf21 cells using RSRHSSYPAGT as substrate assessed as residual enzyme activity at 10 uM measured for 30 mins by [gamma-33P]ATP-based kinase assay | Homo sapiens | 4 | ALA3813662 | cell-based format | Scientific Literature | |
8. | ALA3815559 | Binding | Inhibition of human full length (His)6-tagged Pim-1 expressed in insect Sf21 cells using RSRHSSYPAGT as substrate assessed as residual enzyme activity at 1 uM measured for 30 mins by [gamma-33P]ATP-based kinase assay | Homo sapiens | 4 | ALA3813662 | cell-based format | Scientific Literature | |
9. | ALA3815560 | Binding | Inhibition of human full length (His)6-tagged Pim-1 expressed in insect Sf21 cells using RSRHSSYPAGT as substrate measured for 30 mins by [gamma-33P]ATP-based kinase assay | Homo sapiens | 1 | ALA3813662 | cell-based format | Scientific Literature | |
10. | ALA3815561 | Binding | Inhibition of human full length GST-tagged Pim-2 expressed in Escherichia coli using RSRHSSYPAGT as substrate measured for 30 mins by [gamma-33P]ATP-based kinase assay | Homo sapiens | 1 | ALA3813662 | assay format | Scientific Literature | |
11. | ALA3815562 | Binding | Inhibition of human full length (His)6-tagged Pim-3 expressed in insect Sf21 cells using RSRHSSYPAGT as substrate measured for 30 mins by [gamma-33P]ATP-based kinase assay | Homo sapiens | 1 | ALA3813662 | cell-based format | Scientific Literature | |
12. | ALA3815563 | Binding | Binding affinity to calf thymus double stranded DNA assessed as dsDNA level causing quenching of compound fluorescence by fluorescence spectrophotometric analysis | Bos taurus | 1 | ALA3813662 | nucleic acid format | Scientific Literature | |
13. | ALA3815564 | Binding | Displacement of EtBr from calf thymus double stranded DNA by fluorescence spectrophotometric analysis | Bos taurus | 1 | ALA3813662 | nucleic acid format | Scientific Literature | |
14. | ALA3815581 | Binding | Inhibition of human topoisomerase1 activity at 20 uM using pBR322 plasmid DNA as substrate incubated for 30 mins by EtBr-based gel electrophoresis | Homo sapiens | 1 | ALA3813662 | single protein format | Scientific Literature |