| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3821341 | B | Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor expressed in HEK293 cell membrane assessed as radioligand residence time at 100 uM by microbeta scintillation counting method (Rvb = 61 +/- 4 mins) | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 2. | ALA3821342 | B | Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor expressed in HEK293 cell membrane assessed as radioligand binding at 10 uM by microbeta scintillation counting method relative to control | Homo sapiens | 34 | cell-based format | Scientific Literature | ||
| 3. | ALA3821343 | B | Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane assessed as radioligand binding at 10 uM by microbeta scintillation counting method relative to control | Homo sapiens | 34 | cell-based format | Scientific Literature | ||
| 4. | ALA3821344 | B | Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor expressed in HEK293 cell membrane by microbeta scintillation counting method | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 5. | ALA3821345 | B | Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane by microbeta scintillation counting method | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 6. | ALA3821346 | B | Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane assessed as radioligand residence time at 10 uM by microbeta scintillation counting method (Rvb = 2.8 +/- 0.4 mins) | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 7. | ALA3821347 | B | Ratio of IC50 for human N-terminal FLAG-tagged adenosine A2A receptor expressed in HEK293 cell membrane to IC50 for human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 8. | ALA3821348 | B | Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor expressed in HEK293 cell membrane assessed as decrease in radioligand residence time at 100 uM by microbeta scintillation counting method relative to control | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 9. | ALA3821475 | B | Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane assessed as decrease in radioligand residence time at 10 uM by microbeta scintillation counting method relative to control | Homo sapiens | 5 | cell-based format | Scientific Literature |
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