| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3820761 | A | Inhibition of CYP3A4 in human liver microsomes using midazolam as substrate after 4 mins by LC-MS analysis | Homo sapiens | 11 | tissue-based format | Scientific Literature | ||
| 2. | ALA3820762 | A | Half life in human liver microsomes assessed as CYP-mediated compound degradation at 1 uM by LC-MS analysis | Homo sapiens | 10 | tissue-based format | Scientific Literature | ||
| 3. | ALA3821523 | F | Negative inotropic activity in potassium depolarized guinea pig left atrium assessed as reduction in developed tension at 10'-4 M after 30 mins | Cavia porcellus | 4 | assay format | Scientific Literature | ||
| 4. | ALA3821524 | F | Negative inotropic activity in potassium depolarized guinea pig left atrium assessed as reduction in developed tension after 30 mins | Cavia porcellus | 27 | assay format | Scientific Literature | ||
| 5. | ALA3821527 | F | Negative chronotropic activity in potassium depolarized guinea pig right atrium assessed as reduction in atrial rate at 10'-4 M after 30 mins | Cavia porcellus | 9 | assay format | Scientific Literature | ||
| 6. | ALA3821530 | F | Vasorelaxant activity in potassium depolarized guinea pig aorta assessed as inhibition of calcium-induced contraction at 10'-4 M after 30 mins | Cavia porcellus | 22 | tissue-based format | Scientific Literature | ||
| 7. | ALA3821534 | F | Relaxant activity in potassium depolarized guinea pig ileum longitudinal smooth muscle assessed as inhibition of calcium-induced contraction at 10'-4 M after 30 mins | Cavia porcellus | 4 | tissue-based format | Scientific Literature | ||
| 8. | ALA3821538 | F | Relaxant activity in potassium depolarized guinea pig ileum longitudinal smooth muscle assessed as inhibition of calcium-induced contraction after 30 mins | Cavia porcellus | 9 | tissue-based format | Scientific Literature | ||
| 9. | ALA3821541 | A | Inhibition of CYP2C19 in human liver microsomes using (S)-mephenytoin as substrate after 40 mins by LC-MS analysis | Homo sapiens | 11 | tissue-based format | Scientific Literature | ||
| 10. | ALA3821691 | A | Inhibition of CYP2D6 in human liver microsomes using dextromethorphan as substrate after 10 mins by LC-MS analysis | Homo sapiens | 11 | tissue-based format | Scientific Literature | ||
| 11. | ALA3821692 | A | Intrinsic clearance in human liver microsomes at 1 uM after 2 to 60 mins by LC-MS analysis in presence of NADPH | Homo sapiens | 10 | tissue-based format | Scientific Literature | ||
| 12. | ALA3821693 | A | Stability in human liver microsomes at 1 uM after 2 to 60 mins by LC-MS analysis in absence of NADPH | Homo sapiens | 10 | tissue-based format | Scientific Literature | ||
| 13. | ALA3821694 | A | Inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate after 30 mins by LC-MS analysis | Homo sapiens | 11 | tissue-based format | Scientific Literature | ||
| 14. | ALA3821695 | A | Inhibition of CYP2C9 in human liver microsomes using tolbutamide as substrate after 20 mins by LC-MS analysis | Homo sapiens | 11 | tissue-based format | Scientific Literature | ||
| 15. | ALA3821882 | A | Inhibition of CYP3A4 in human liver microsomes using testosterone as substrate after 5 mins by LC-MS analysis | Homo sapiens | 11 | tissue-based format | Scientific Literature |
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