| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3830343 | B | Agonist activity at Gal4-tagged human PPAR-alpha expressed in HEK cells by transactivation assay | Homo sapiens | 18 | ALA3826929 | cell-based format | Scientific Literature | |
| 2. | ALA3830344 | B | Agonist activity at Gal4-tagged human PPAR-gamma expressed in HEK cells by transactivation assay | Homo sapiens | 18 | ALA3826929 | cell-based format | Scientific Literature | |
| 3. | ALA3830345 | B | Selectivity ratio of EC50 for Gal4-tagged human PPAR-gamma expressed in HEK cells to EC50 for Gal4-tagged human PPAR-alpha expressed in HEK cells | Homo sapiens | 17 | ALA3826929 | cell-based format | Scientific Literature | |
| 4. | ALA3830346 | B | Binding affinity to human GST-tagged PPAR-alpha LBD expressed in Escherichia coli BL21 (DE3) PlysS after 30 mins in presence of fluorescein ligand FLA-A by fluorescence polarization assay | Homo sapiens | 4 | ALA3826929 | assay format | Scientific Literature | |
| 5. | ALA3830347 | B | Binding affinity to human GST-tagged PPAR-gamma LBD expressed in Escherichia coli BL21 after 30 mins in presence of fluorescein ligand FLA-A by fluorescence polarization assay | Homo sapiens | 4 | ALA3826929 | assay format | Scientific Literature | |
| 6. | ALA3830348 | A | Tmax in Balb/c mouse at 10 mg/kg, po | Mus musculus | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 7. | ALA3830349 | A | Tmax in Sprague-Dawley rat at 8 mg/kg, po | Rattus norvegicus | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 8. | ALA3830447 | A | Tmax in dog at 2 mg/kg, po | Canis lupus familiaris | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 9. | ALA3830448 | A | Tmax in cynomolgus monkey at 2 mg/kg, po | Macaca fascicularis | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 10. | ALA3830449 | A | Cmax in Balb/c mouse at 10 mg/kg, po | Mus musculus | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 11. | ALA3830450 | A | Cmax in Sprague-Dawley rat at 8 mg/kg, po | Rattus norvegicus | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 12. | ALA3830451 | A | Cmax in dog at 2 mg/kg, po | Canis lupus familiaris | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 13. | ALA3830452 | A | Cmax in cynomolgus monkey at 2 mg/kg, po | Macaca fascicularis | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 14. | ALA3830453 | A | AUC (0 to 8 hrs) in Balb/c mouse at 5 mg/kg, iv | Mus musculus | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 15. | ALA3830454 | A | AUC (0 to 8 hrs) in Balb/c mouse at 10 mg/kg, po | Mus musculus | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 16. | ALA3830455 | A | AUC (0 to 8 hrs) in Sprague-Dawley rat at 4 mg/kg, iv | Rattus norvegicus | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 17. | ALA3830456 | A | AUC (0 to 8 hrs) in Sprague-Dawley rat at 8 mg/kg, po | Rattus norvegicus | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 18. | ALA3830457 | A | AUC (0 to 8 hrs) in dog at 1 mg/kg, iv | Canis lupus familiaris | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 19. | ALA3830458 | A | AUC (0 to 8 hrs) in dog at 2 mg/kg, po | Canis lupus familiaris | 1 | ALA3826929 | organism-based format | Scientific Literature | |
| 20. | ALA3830459 | A | AUC (0 to 8 hrs) in cynomolgus monkey at 1 mg/kg, iv | Macaca fascicularis | 1 | ALA3826929 | organism-based format | Scientific Literature |
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