# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3863850 | B | Displacement of [3H]WAY100635 from human 5-HT1AR expressed in CHO cell membranes at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | cell-based format | Scientific Literature | |
2. | ALA3863851 | B | Displacement of [3H]5-CT from human 5-HT1BR expressed in HEK cell membranes at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | cell-based format | Scientific Literature | |
3. | ALA3863852 | B | Displacement of [3H]5-CT from human 5-HT1D receptor expressed in HEK-T cell membranes at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | cell-based format | Scientific Literature | |
4. | ALA3863853 | B | Displacement of [3H]5-HT from human 5-HT1E receptor expressed in HEK cell membranes at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | cell-based format | Scientific Literature | |
5. | ALA3863854 | B | Displacement of [3H]GR113808 from human 5-HT4 receptor at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | single protein format | Scientific Literature | |
6. | ALA3863855 | B | Displacement of [3H]LSD from human 5-HT6 receptor expressed in HEK cell membranes at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | cell-based format | Scientific Literature | |
7. | ALA3863856 | B | Displacement of [3H]LSD from human 5-HT7A receptor expressed in HEK cell membranes at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | cell-based format | Scientific Literature | |
8. | ALA3863857 | B | Displacement of [3H]GR65630 from human 5-HT3 receptor expressed in HEK-T cell membranes at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 32 | ALA3862033 | cell-based format | Scientific Literature | |
9. | ALA3863858 | B | Displacement of [3H]LSD from human 5-HT5A receptor expressed in Flp-In-CHO cell membranes incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | cell-based format | Scientific Literature | |
10. | ALA3863859 | B | Displacement of [3H]ketanserin from human 5-HT2A receptor expressed in HEK-T cell membranes at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | cell-based format | Scientific Literature | |
11. | ALA3863860 | B | Displacement of [3H]lysergic from human 5-HT2BR expressed in HEK cell membranes incubated in dark for 90 mins by microbeta scintillation counting method | Homo sapiens | 27 | ALA3862033 | cell-based format | Scientific Literature | |
12. | ALA3863861 | B | Displacement of [3H]lysergic from human 5-HT2BR expressed in HEK cell membranes at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | cell-based format | Scientific Literature | |
13. | ALA3863862 | B | Displacement of [3H]mesulergine from human 5-HT2CR expressed in Flp-In HEK cell membranes incubated for 90 mins under dark condition by microbeta scintillation counting method | Homo sapiens | 26 | ALA3862033 | cell-based format | Scientific Literature | |
14. | ALA3863863 | B | Displacement of [3H]mesulergine from human 5-HT2CR expressed in Flp-In HEK cell membranes at 10 uM incubated for 90 mins under dark condition by microbeta scintillation counting method relative to control | Homo sapiens | 33 | ALA3862033 | cell-based format | Scientific Literature | |
15. | ALA3863864 | B | Displacement of [3H]N6-phenylisopropyladenosine from recombinant human A1AR expressed in CHO cell membranes after 60 mins by liquid scintillation counting method | Homo sapiens | 21 | ALA3862033 | cell-based format | Scientific Literature | |
16. | ALA3863867 | B | Displacement of [3 H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from recombinant human adenosine receptor A2A expressed in HEK293 cell membranes after 60 mins by liquid scintillation counting method | Homo sapiens | 14 | ALA3862033 | cell-based format | Scientific Literature | |
17. | ALA3863870 | B | Displacement of [125l]N 6-(4-amino-3-iodobenzyl)adenosine-5'-N-methyluronamide from recombinant human A3AR expressed in CHO cell membranes after 60 mins by gamma counting method | Homo sapiens | 24 | ALA3862033 | cell-based format | Scientific Literature | |
18. | ALA3863872 | B | Selectivity ratio of Ki for human 5-HT2CR expressed in Flp-In HEK cell membranes to Ki for human 5-HT2B expressed in HEK cell membranes | Homo sapiens | 3 | ALA3862033 | cell-based format | Scientific Literature | |
19. | ALA3863875 | F | Agonist activity at recombinant human A1AR expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation at 10 uM after 15 mins relative to N6-cyclopentyladenosine | Homo sapiens | 2 | ALA3862033 | cell-based format | Scientific Literature | |
20. | ALA3863877 | F | Antagonist activity at human 5-HT2BR expressed in Flp-In HEK cells assessed as inhibition of 5-HT-induced calcium mobilization preincubated for 5 to 10 mins followed 5-HT addition by Fluo-4 dye based FLIPR assay | Homo sapiens | 6 | ALA3862033 | cell-based format | Scientific Literature |