| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3880754 | Binding | Antagonist activity at rat alpha1B N-type calcium channel expressed in HEK293 cells assessed as 0.067 Hz current frequency dependent channel blocking for 2 mins in presence of Ba2+ by whole-cell patch clamp assay | Rattus norvegicus | 33 | ALA3880396 | cell-based format | Patent Bioactivity Data | |
| 2. | ALA3880755 | Binding | Antagonist activity at rat alpha1B N-type Ca2+ channel expressed in HEK293 cells assessed as 0.2 Hz current frequency dependent channel blocking for 2 mins in presence of Ba2+ by whole-cell patch clamp assay | Rattus norvegicus | 33 | ALA3880396 | cell-based format | Patent Bioactivity Data | |
| 3. | ALA3880756 | Binding | Antagonist activity at rat brain alpha1B/alpha2b/beta1b N-type calcium channel expressed in HEK293 cells assessed as 0.1 Hz current frequency dependent channel blocking for 2 to 3 mins in presence of Ba2+ by whole-cell patch clamp assay | Rattus norvegicus | 6 | ALA3880396 | cell-based format | Patent Bioactivity Data | |
| 4. | ALA3880757 | Binding | Antagonist activity at alpha1C/alpha2delta/beta1b L-type calcium channel (unknown origin) expressed in HEK293 cells assessed as 0.1 Hz current frequency dependent channel blocking for 2 to 3 mins in presence of Ba2+ by whole-cell patch clamp assay | Homo sapiens | 6 | ALA3880396 | cell-based format | Patent Bioactivity Data | |
| 5. | ALA3880758 | Binding | Antagonist activity at alpha1A/alpha2delta/beta1b P/Q-type calcium channel (unknown origin) expressed in HEK293 cells assessed as 0.1 Hz current frequency dependent channel blocking for 2 to 3 mins in presence of Ba2+ by whole-cell patch clamp assay | Homo sapiens | 6 | ALA3880396 | cell-based format | Patent Bioactivity Data | |
| 6. | ALA3880759 | Binding | Selectivity ratio of IC50 for alpha1A/alpha2delta/beta1b P/Q-type calcium channel (unknown origin) to IC50 for rat brain alpha1B/alpha2b/beta1b N-type calcium channel | 6 | ALA3880396 | assay format | Patent Bioactivity Data | ||
| 7. | ALA3880760 | Binding | Selectivity ratio of IC50 for alpha1C/alpha2delta/beta1b L-type calcium channel (unknown origin) to IC50 for rat brain alpha1B/alpha2b/beta1b N-type calcium channel | 6 | ALA3880396 | assay format | Patent Bioactivity Data |
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