| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3869635 | A | Clearance in rhesus monkey at 1 mg/kg, iv or 2 mg/kg, po administered qd | Macaca mulatta | 1 | organism-based format | Scientific Literature | ||
| 2. | ALA3869636 | A | Stability in dog microsomes assessed as compound remaining at 45 mins | Canis lupus familiaris | 1 | assay format | Scientific Literature | ||
| 3. | ALA3869637 | A | Stability in human hepatocytes assessed as compound remaining at 90 mins | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA3869638 | A | Inhibition of CYP2C9 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 5. | ALA3869639 | A | Stability in rhesus monkey hepatocytes assessed as compound remaining at 90 mins | Macaca mulatta | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA3869640 | A | Stability in human microsomes assessed as compound remaining at 45 mins | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 7. | ALA3869641 | A | Stability in rhesus monkey microsomes assessed as compound remaining at 45 mins | Macaca mulatta | 1 | assay format | Scientific Literature | ||
| 8. | ALA3869642 | A | Stability in rat microsomes assessed as compound remaining at 45 mins | Rattus norvegicus | 1 | assay format | Scientific Literature | ||
| 9. | ALA3869647 | B | Inhibition of human ROMK expressed in CHO cells after 6 mins at -70 mV holding potential by electrophysiology method | Homo sapiens | 28 | cell-based format | Scientific Literature | ||
| 10. | ALA3869650 | B | Inhibition of human ERG by electrophysiology method | Homo sapiens | 22 | single protein format | Scientific Literature | ||
| 11. | ALA3869651 | B | Selectivity ratio of IC50 for human ERG by electrophysiology method to IC50 for human ROMK expressed in CHO cells | Homo sapiens | 22 | cell-based format | Scientific Literature | ||
| 12. | ALA3869652 | B | Inhibition of Kir7.1 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA3869653 | B | Inhibition of Kir2.1 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA3869654 | B | Inhibition of Kir4.1 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA3869655 | B | Inhibition of Nav1.5 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA3869656 | B | Inhibition of Cav1.2 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA3869657 | B | Inhibition of Somatostatin receptor type 2 (unknown origin) at 10 uM by radioligand binding assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA3869658 | B | Inhibition of Somatostatin receptor type 2 (unknown origin) by radioligand binding assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA3869659 | B | Selectivity ratio of IC50 for Somatostatin receptor type 2 (unknown origin) to IC50 for human ROMK expressed in CHO cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA3869660 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature |
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