| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3878974 | B | Inhibition of human BCR/ABL p210 fusion protein expressed in BAF3 cells assessed as growth inhibition measured after 72 hrs by CellTiter-Glo or CCK8 assay | Homo sapiens | 30 | cell-based format | Scientific Literature | ||
| 2. | ALA3878975 | B | Inhibition of Tel-fused c-KIT (unknown origin) expressed in BAF3 cells assessed as growth inhibition measured after 72 hrs by CellTiter-Glo or CCK8 assay | Homo sapiens | 30 | cell-based format | Scientific Literature | ||
| 3. | ALA3878976 | A | Growth inhibition of mouse BAF3 cells measured after 72 hrs by CellTiter-Glo or CCK8 assay | Mus musculus | 30 | cell-based format | Scientific Literature | ||
| 4. | ALA3878977 | B | Inhibition of C-terminal His-tagged human ABL1 expressed in baculovirus infected SF9 cells using Tyr 02 peptide as substrate measured after 1 hr by FRET based Z'Lyte assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 5. | ALA3878978 | B | Inhibition of recombinant C-terminal polyhistidine-tagged human c-KIT expressed in mammalian expression system using Tyr 06 peptide as substrate measured after 1hr by FRET based Z'Lyte assay | Homo sapiens | 6 | assay format | Scientific Literature | ||
| 6. | ALA3878979 | B | Inhibition of C-terminal His-tagged human ABL1 expressed in baculovirus infected SF9 cells assessed as residual activity at 1 uM using Tyr 02 peptide as substrate measured after 1 hr by FRET based Z'Lyte assay relative to control | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA3878980 | B | Inhibition of recombinant C-terminal polyhistidine-tagged human c-KIT expressed in mammalian expression system assessed as residual activity at 1 uM using Tyr 06 peptide as substrate measured after 1hr by FRET based Z'Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 8. | ALA3878981 | B | Inhibition of recombinant C-terminal His-tagged human LCK cytoplasmic domain expressed in baculovirus expression system assessed as residual activity at 1 uM measured after 1 hr by FRET based Z'Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA3878982 | B | Inhibition of full length recombinant His-tagged human BLK cytoplasmic domain expressed in baculovirus expression system assessed as residual activity at 1 uM measured after 1 hr by FRET based Z'Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA3878983 | B | Inhibition of full length recombinant His-tagged human BLK cytoplasmic domain expressed in baculovirus expression system measured after 1 hr by FRET based Z'Lyte assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA3878984 | B | Inhibition of recombinant His-tagged human CSF1R cytoplasmic domain expressed in baculovirus expression system assessed as residual activity at 1 uM measured after 1 hr by FRET based Z'Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA3878985 | B | Inhibition of recombinant His-tagged human CSF1R cytoplasmic domain expressed in baculovirus expression system measured after 1 hr by FRET based Z'Lyte assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA3878986 | B | Inhibition of human GST-tagged DDR1 cytoplasmic domain expressed in baculovirus expression system assessed as residual activity at 1 uM measured after 1 hr by FRET based Z'Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA3878987 | B | Inhibition of human GST-tagged DDR1 cytoplasmic domain expressed in baculovirus expression system measured after 1 hr by FRET based Z'Lyte assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA3878988 | B | Inhibition of recombinant His-tagged human DDR2 cytoplasmic domain expressed in baculovirus expression system assessed as residual activity at 1 uM measured after 1 hr by FRET based Z'Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA3878989 | B | Inhibition of recombinant His-tagged human DDR2 cytoplasmic domain expressed in baculovirus expression system measured after 1 hr by FRET based Z'Lyte assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA3878990 | B | Inhibition of recombinant C-terminal His-tagged human LCK cytoplasmic domain expressed in baculovirus expression system measured after 1 hr by FRET based Z'Lyte assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA3878991 | B | Inhibition of LOK (unknown origin) assessed as residual activity at 1 uM measured after 1 hr by FRET based Z'Lyte assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA3878992 | B | Inhibition of LOK (unknown origin) measured after 1 hr by FRET based Z'Lyte assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA3878993 | B | Inhibition of recombinant His-tagged human PDGFR-beta cytoplasmic domain (558 to 1106 residues) expressed in baculovirus expression system assessed as residual activity at 1 uM measured after 1 hr by FRET based Z'Lyte assay relative to control | Homo sapiens | 1 | assay format | Scientific Literature |
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