| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3855716 | B | Transactivation of ProLink tagged human PPARdelta transfected in CHO-K1 cells assessed as interaction with EA labelled SRCP after 3 to 16 hrs by beta galactosidase reporter gene assay | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 2. | ALA3855717 | B | Transactivation of human Gal4-PPARdelta LBD transfected in African green monkey CV1 cells after 24 hrs by luciferase reporter gene assay | Homo sapiens | 9 | cell-based format | Scientific Literature | ||
| 3. | ALA4181577 | B | Transactivation of yeast GAL4 DNA binding domain-fused PPARdelta LBD (unknown origin) expressed in CV-1 cells after 24 hrs by luciferase reporter gene assay | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 4. | ALA4181578 | B | Activation of human PPARdelta LBD expressed in CHO-K1 cells by beta galactosidase enzyme fragment complement based fluorescence assay | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
| 5. | ALA4181579 | A | Half life in CD-1 mouse at 3 mg/kg, iv | Mus musculus | 12 | organism-based format | Scientific Literature | ||
| 6. | ALA4181580 | A | Clearance in CD-1 mouse at 3 mg/kg, iv | Mus musculus | 13 | organism-based format | Scientific Literature | ||
| 7. | ALA4181581 | A | AUC in CD-1 mouse at 3 mg/kg, iv | Mus musculus | 12 | organism-based format | Scientific Literature | ||
| 8. | ALA4181582 | B | Activation of human PPARalpha LBD expressed in CHO-K1 cells by beta galactosidase enzyme fragment complement based fluorescence assay | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 9. | ALA4181583 | B | Transactivation of yeast GAL4 DNA binding domain-fused PPARalpha LBD (unknown origin) expressed in CV-1 cells after 24 hrs by luciferase reporter gene assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 10. | ALA4181584 | B | Activation of human PPARgamma LBD expressed in CHO-K1 cells by beta galactosidase enzyme fragment complement based fluorescence assay | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 11. | ALA4181585 | B | Transactivation of yeast GAL4 DNA binding domain-fused PPARgamma LBD (unknown origin) expressed in CV-1 cells after 24 hrs by luciferase reporter gene assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 12. | ALA4181586 | B | Binding affinity to His-tagged PPARdelta (unknown origin) by SPR assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA4181587 | P | Thermodynamic solubility of the compound | 1 | small-molecule physicochemical format | Scientific Literature | |||
| 14. | ALA4181588 | A | Efflux ratio of permeability in human Caco2 cells | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA4181589 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA4181590 | A | Inhibition of CYP2C9 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA4181591 | A | Inhibition of CYP2C19 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA4181592 | A | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA4181593 | A | Inhibition of CYP1A2 (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA4181594 | A | Half life in CD-1 mouse at 1 mg/kg, iv | Mus musculus | 1 | organism-based format | Scientific Literature |
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