# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3880925 | B | Inhibition of HDAC (unknown origin) using Fluor-Lys as substrate | Homo sapiens | 20 | ALA3880414 | protein format | Patent Bioactivity Data | |
2. | ALA3880928 | F | Antiproliferative activity against human SQ20B cells | Homo sapiens | 17 | ALA3880414 | cell-based format | Patent Bioactivity Data | |
3. | ALA3880929 | F | Antiproliferative activity against human PC3 cells | Homo sapiens | 17 | ALA3880414 | cell-based format | Patent Bioactivity Data | |
4. | ALA3880930 | F | Antiproliferative activity against human MCF7 cells | Homo sapiens | 17 | ALA3880414 | cell-based format | Patent Bioactivity Data | |
5. | ALA3880931 | F | Antiproliferative activity against human HeLa cells | Homo sapiens | 17 | ALA3880414 | cell-based format | Patent Bioactivity Data | |
6. | ALA3880939 | B | Inhibition of HDAC1 in human HeLa cell nuclear extracts assessed as residual activity at 0.5 uM relative to control | Homo sapiens | 16 | ALA3880414 | cell-based format | Patent Bioactivity Data | |
7. | ALA3880940 | B | Inhibition of HDAC2 in human HeLa cell nuclear extracts assessed as residual activity at 0.5 uM relative to control | Homo sapiens | 16 | ALA3880414 | cell-based format | Patent Bioactivity Data | |
8. | ALA3880941 | B | Inhibition of HDAC3 in human HeLa cell nuclear extracts assessed as residual activity at 0.5 uM relative to control | Homo sapiens | 16 | ALA3880414 | cell-based format | Patent Bioactivity Data | |
9. | ALA3880942 | B | Inhibition of HDAC8 (unknown origin) assessed as residual activity at 0.5 uM relative to control | Homo sapiens | 16 | ALA3880414 | single protein format | Patent Bioactivity Data | |
10. | ALA5226443 | B | Inhibition of human HDAC1 using FAM-labeled acetylated peptide as substrate incubated for 17 hrs by fluorescence based assay | Homo sapiens | 4 | ALA5226279 | single protein format | Scientific Literature | |
11. | ALA5226444 | B | Inhibition of human HDAC2 using FAM-labeled acetylated peptide as substrate incubated for 17 hrs by fluorescence based assay | Homo sapiens | 4 | ALA5226279 | single protein format | Scientific Literature | |
12. | ALA5226445 | B | Inhibition of human HDAC8 using FAM-labeled acetylated peptide as substrate incubated for 17 hrs by fluorescence based assay | Homo sapiens | 4 | ALA5226279 | single protein format | Scientific Literature | |
13. | ALA5226446 | B | Inhibition of human HDAC6 using FAM-labeled acetylated peptide as substrate incubated for 17 hrs by fluorescence based assay | Homo sapiens | 4 | ALA5226279 | single protein format | Scientific Literature | |
14. | ALA5226447 | B | Inhibition of human HDAC10 using FAM-labeled acetylated peptide as substrate incubated for 17 hrs by fluorescence based assay | Homo sapiens | 4 | ALA5226279 | single protein format | Scientific Literature | |
15. | ALA5226448 | B | Selectivity index, ratio of IC50 for inhibition of human HDAC1 to IC50 for inhibition of human HDAC6 | Homo sapiens | 4 | ALA5226279 | assay format | Scientific Literature |